Targeted α-therapy using astatine ( 211 At)-labeled PSMA1, 5, and 6: a preclinical evaluation as a novel compound.
Tadashi WatabeKazuko Kaneda-NakashimaYoshifumi ShirakamiYuichiro KadonagaKazuhiro OoeYang WangHiromitsu HabaAtsushi ToyoshimaJens CardinaleFrederik L GieselNoriyuki TomiyamaKoichi FukasePublished in: European journal of nuclear medicine and molecular imaging (2022)
At]PSMA5 should be considered a new possible TAT for metastatic CRPC, and translational prospective trials are warranted.