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Brain pharmacokinetics of two BBB penetrating bispecific antibodies of different size.

Rebecca FaresjöGillian BonviciniXiaotian T FangXimena AguilarDag SehlinStina Syvanen
Published in: Fluids and barriers of the CNS (2021)
A smaller size and lower TfR1 avidity are likely important for fast parenchymal delivery, while elimination of brain-associated bispecific antibodies may not be dependent on these characteristics.
Keyphrases
  • resting state
  • white matter
  • functional connectivity
  • blood brain barrier
  • cerebral ischemia
  • brain injury
  • subarachnoid hemorrhage