Anodic dearomatization of 2-alkynylanilines for the synthesis of multi-functionalized indoles.
Zhuowen ChenQiuqin HeHao GuoRenhua FanPublished in: Chemical communications (Cambridge, England) (2022)
An anodic oxidative dearomatization reaction of 2-alkynylanilines was developed. The formed dearomatized compounds were used as versatile precursors in the synthesis of a variety of benzenoid ring multi-functionalized indoles through simple conversions.
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