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Hits and misses with animal models of narcolepsy and the implications for drug discovery.

Ramakrishna NirogiPradeep JayarajanVijay BenadeRenny AbrahamVinod Kumar Goyal
Published in: Expert opinion on drug discovery (2024)
Research in canine and mouse models have linked narcolepsy to the O×R2mutation and orexin deficiency, leading to new diagnostic criteria and a drug development focus. Advancements in pharmacological therapies have significantly improved narcolepsy management, with insights from both clinical experience and from animal models having led to new treatments such as low sodium oxybate and solriamfetol. However, challenges persist in addressing symptoms beyond excessive daytime sleepiness and cataplexy, highlighting the need for further research, including the development of diurnal animal models to enhance understanding and treatment options for narcolepsy.
Keyphrases
  • drug discovery
  • sleep quality
  • obstructive sleep apnea
  • mouse model
  • weight gain
  • depressive symptoms
  • sleep apnea
  • physical activity
  • replacement therapy