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A Bifunctional Ligand Enables Gold-Catalyzed Hydroarylation of Terminal Alkynes under Soft Reaction Conditions.

Ting LiYuhan YangBaomin LuoBo LiLuyi ZongWeiguang KongHao YangXinpeng ChengLiming Zhang
Published in: Organic letters (2020)
An efficient gold-catalyzed hydroarylation of alkynes under soft reaction conditions is developed by utilizing a bifunctional ligand. This transformation features a broad substrate scope and thus exhibits moderate to excellent efficiency.
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