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Palladium-Catalyzed Enantioselective Decarboxylative Allylic Alkylation of Protected Benzoin-Derived Enol Carbonates.

Rémi LavernheEric J AlexyHaiming ZhangBrian M Stoltz
Published in: Advanced synthesis & catalysis (2019)
The enantioselective palladium-catalyzed decarboxylative allylic alkylation of fully substituted α-hydroxy acyclic enol carbonates providing tetrasubstituted benzoin derivatives is reported. Investigation into the transformation revealed that preparation of the starting material as a single enolate isomer is crucial for optimal enantioselectivity. The obtained alkylation products contain multiple reactive sites that can be utilized toward the synthesis of stereochemically rich derivatives. COMMUNICATION.
Keyphrases
  • visible light
  • structure activity relationship
  • molecular docking
  • single cell
  • tandem mass spectrometry