Lewis Acid-Facilitated Radiofluorination of MN3PU: A LRRK2 Radiotracer.
Noeen MalikShreya BendreRalf SchirrmacherPaul SchafferPublished in: Molecules (Basel, Switzerland) (2020)
RCYs of [18F]FMN3PU (7) improved from ~5% using conventional nucleophilic radiofluorination, up to 41 ± 1% using Lewis-acid supported SNAr.