Copper-Catalyzed Decarboxylative Cycloaddition of Propiolic Acids, Azides, and Arylboronic Acids: Construction of Fully Substituted 1,2,3-Triazoles.
Xiang-Xiang WangYangchun XinYi LiWen-Jin XiaBin ZhouRui-Rong YeYa-Min LiPublished in: The Journal of organic chemistry (2020)
A copper-catalyzed decarboxylative cycloaddition of propiolic acids, azides, and arylboronic acids is described. The present reaction provides an efficient and convenient method for the synthesis of various fully substituted 1,2,3-triazoles from readily available starting materials. A possible mechanism is proposed.
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