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A Highly Stereoselective Redox Isomerization-Reductive Deuteration Sequence of Propargyl Amines to α-Deuterated Amino Acids.

Zhipeng ZhaoHongrui LinZheng ZhangXiaotong GaoCongbin JiJian ZhouFeng Zhou
Published in: Organic letters (2023)
Herein, we report a Cu-catalyzed redox isomerization-reductive deuteration sequence, providing facile access to a range of α-deuterated amino acid esters featuring an Z -configured alkene moiety with high yields. The advantages of this sequence include mild conditions, broad substrate scope, and excellent stereoselectivity. This research also represents a rare example of the Z -selective redox isomerization of propargyl amines.
Keyphrases
  • amino acid
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  • highly efficient
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  • structural basis