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Nitrogen-Containing 2,3-Dihydroquinazolinone Compounds as Na v 1.8 Inhibitors for Treating Pain and Cardiovascular Diseases.

Rachel Mata
Published in: ACS medicinal chemistry letters (2023)
Provided herein are novel nitrogen-containing 2,3-dihydroquinazolinone compounds as Na v 1.8 inhibitors, pharmaceutical compositions, use of such compounds in treating pain and cardiovascular diseases, and processes for preparing such compounds.
Keyphrases
  • cardiovascular disease
  • chronic pain
  • pain management
  • neuropathic pain
  • type diabetes
  • spinal cord injury
  • coronary artery disease
  • postoperative pain