Pharmacokinetic and pharmacodynamic assessment of histamine H3 receptor occupancy by enerisant: a human PET study with a novel H3 binding ligand, [11C]TASP457.
Yasuyuki KimuraKeisuke TakahataToshiharu ShimazakiSoichiro KitamuraChie SekiYoko IkomaMasanori IchiseKazunori KawamuraMakiko YamadaMing-Rong ZhangMakoto HiguchiIzumi NishinoTetsuya SuharaPublished in: European journal of nuclear medicine and molecular imaging (2021)
This study was retrospectively registered with ClinicalTrials.gov (NCT04631276) on November 17, 2020.