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Pharmacokinetic and pharmacodynamic assessment of histamine H3 receptor occupancy by enerisant: a human PET study with a novel H3 binding ligand, [11C]TASP457.

Yasuyuki KimuraKeisuke TakahataToshiharu ShimazakiSoichiro KitamuraChie SekiYoko IkomaMasanori IchiseKazunori KawamuraMakiko YamadaMing-Rong ZhangMakoto HiguchiIzumi NishinoTetsuya Suhara
Published in: European journal of nuclear medicine and molecular imaging (2021)
This study was retrospectively registered with ClinicalTrials.gov (NCT04631276) on November 17, 2020.
Keyphrases
  • endothelial cells
  • computed tomography
  • pet ct
  • clinical evaluation