Halogen Replacement on the Lysine Side Chain of Lys-Urea-Glu-Based PSMA Inhibitors Leads to Significant Changes in Targeting Properties.
Li XiaYang LiuPing CaiYue FengHongmei YuanSufan TangYin Wen WangNan LiuYue ChenZhijun ZhouPublished in: Molecular imaging and biology (2023)
Ga]Ga-DOTA-SC691-R to PSMA. The bulkier and less electronegative Br (or I) elements are preferred for structural modifications here.