Pd-Catalyzed Aryl C-H Amination with Diaziridinone.

This work describes an efficient Pd-catalyzed ortho -C-H amination of N -(quinolin-8-yl)benzamides with di- t -butyldiaziridinone, providing a variety of anthranilic amides in good yields. The reaction likely involves the formation of a pallada(II)heterocycle via aryl C-H activation and subsequent amination with di- t -butyldiaziridinone.