Organotrifluoroborate enhances tumor targeting of fibroblast activation protein inhibitors for targeted radionuclide therapy.
Yu LiuHaocheng TangTianchi SongMengxin XuJunyi ChenXi-Yang CuiYuxiang HanZhu LiZhibo LiuPublished in: European journal of nuclear medicine and molecular imaging (2023)
The organotrifluoroborate linker may be of importance to optimize FAP-targeted radiopharmaceuticals, and the short half-lived α-emitters may be of choice for the rapid-cleared small molecule-based radiopharmaceuticals.