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A Minimal PBPK Model for Plasma and Cerebrospinal Fluid Pharmacokinetics of Trastuzumab after Intracerebroventricular Administration in Patients with HER2-Positive Brain Metastatic Localizations.

Alicja PuszkielGuilhem BousquetFrançoise Stanke-LabesqueJeanick StoccoPhilippe DecqLucie ChevillardStéphane GoutagnyXavier Declèves
Published in: Pharmaceutical research (2023)
Continuous icv infusion of trastuzumab at 1.0 mg/h could be an alternative dosing regimen to rapidly achieve intraventricular CSF therapeutic concentrations.
Keyphrases
  • cerebrospinal fluid
  • epidermal growth factor receptor
  • metastatic breast cancer
  • small cell lung cancer
  • squamous cell carcinoma
  • white matter
  • low dose
  • resting state
  • multiple sclerosis
  • blood brain barrier