Importance of receptor expression in the classification of novel ligands at the M 2 muscarinic acetylcholine receptor.
Ye JiangMahmuda YeasminArisbel B GondinArthur ChristopoulosCeline ValantWessel A C BurgerDavid M ThalPublished in: British journal of pharmacology (2022)
bias of compounds 6A and 7A highlighting the importance of cellular background when classifying new ligands.