Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18 F-fluorination of boroxines, in vitro and initial in vivo evaluation.
Kim-Viktoria BolikJan HellmannSimone MaschauerEduard NeuJürgen EinsiedelPatrick RissNora VoggJörg KönigMartin F FrommHarald HübnerPeter GmeinerOlaf PrantePublished in: EJNMMI research (2024)
F]1f provide a solid basis for further development of suitable OXR PET ligands for brain imaging.