Palladium-Mediated Site-Selective C-H Radio-iodination.
Emmanuelle DubostVictor BabinFlorian BenoistAlexandra HébertPierre BarbeyCéline CholletJean-Philippe BouillonAlain ManriqueGrégory PietersFrédéric FabisThomas CaillyPublished in: Organic letters (2018)
The palladium-mediated C-H radio-iodination of arenes using sodium iodide as the primary isotopic source is reported and performed without chemical know-how in 30 min and applied to the synthesis of complex radio-iodinated compounds of biological interest.
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