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Rational Drug Discovery for Isoxazole Based VEGFR2 Inhibition.

Shital M PatilIndrani MahadikShashikant V BhandariKalyani D AsgaonkarVrushali D RandiveAishwarya M Edake
Published in: Current drug discovery technologies (2024)
According to QSAR studies, more electron-donating groups on the benzene ring linked to the isoxazole were shown to be necessary for activity. In molecular docking studies, most compounds have shown stronger affinity for the crucial amino acids Cys:919, Asp:1046, and Glu:885, which are found in typical drugs. All NCEs passed the Lipinski screening.
Keyphrases
  • molecular docking
  • drug discovery
  • molecular dynamics simulations
  • amino acid
  • case control
  • vascular endothelial growth factor
  • molecular dynamics
  • structure activity relationship