Development of a practical synthesis of etravirine via a microwave-promoted amination.
Da FengFenju WeiZhao WangDongwei KangPeng ZhanXinyong LiuPublished in: Chemistry Central journal (2018)
Overall, we developed a practical synthesis of ETV via a microwave-promoted method, and the synthetic procedure could be amenable to scale-up, and production costs could be significantly lowered.