Proof of pharmacology of Org 48775-0, a p38 MAP kinase inhibitor, in healthy volunteers.
Matthijs MoerlandAndrea J KalesKaren BroekhuizenUlla NässanderRob NelissenMarieke L de KamPierre A M PeetersJacobus BurggraafPublished in: British journal of clinical pharmacology (2020)
Org 48,775-0 has the capacity to significantly inhibit MAP kinase activity in humans without safety concerns.