SAR Studies of the Leupyrrins: Design and Total Synthesis of Highly Potent Simplified Leupylogs.

Paul R WosniokChristopher KnopfSandra DreisigackerJ Manuel Orozco-RodriguezBettina HinkelmannPeter P MuellerMark BrönstrupDirk Menche

Published in: Chemistry (Weinheim an der Bergstrasse, Germany) (2020)

Invited for the cover of this issue is the group of Dirk Menche at the University of Bonn. The image depicts the natural product leupyrrin A1 and a synthetic leupylog in balance on an IC50 weighing scale. Read the full text of the article at 10.1002/chem.202002622.

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