Selectivity, cell permeability and oral availability studies of novel bromophenol derivative HPN as protein tyrosine phosphatase 1B inhibitor.
Jiao LuoQi XuBo JiangRenshuai ZhangXiaoling JiaXiangqian LiLijun WangChuanlong GuoNing WuDayong ShiPublished in: British journal of pharmacology (2017)
Our results indicate that HPN is a specific PTP1B inhibitor, with anti-diabetic properties and good cell permeability and oral availability.