The polar warhead of a TRIM24 bromodomain inhibitor rearranges a water-mediated interaction network.
Jiuyang LiuFudong LiHongyu BaoYiyang JiangShuya ZhangRongsheng MaJia GaoJihui WuKe RuanPublished in: The FEBS journal (2017)
Structural data are available in the PDB under the accession numbers 5H1T, 5H1U, and 5H1V.