Benjamin R Bellenie

ORCID

Publication Activity (10 Years)

Years Active: 2020-2024
Publications (10 Years): 13

Top Venues

Journal of medicinal chemistry

ACS chemical biology

This page only lists publications with an associated author ORCID identifier.

Publications

Katie L Thomas, Habib Bouguenina, Daniel S J Miller, Fernando J Sialana, Thomas G Hayhow, Jyoti S Choudhary, Olivia W Rossanese, Benjamin R Bellenie
Degradation by Design: New Cyclin K Degraders from Old CDK Inhibitors. ACS chemical biology 19 (1) (2024)
Katie L Thomas, Habib Bouguenina, Daniel S J Miller, Fernando J Sialana, Thomas G Hayhow, Jyoti S Choudhary, Olivia W Rossanese, Benjamin R Bellenie
Degradation by Design: New Cyclin K Degraders from Old CDK Inhibitors. ACS chemical biology (2024)
Katie L Thomas, Habib Bouguenina, Daniel S J Miller, Fernando J Sialana, Thomas G Hayhow, Jyoti S Choudhary, Olivia W Rossanese, Benjamin R Bellenie
Degradation by Design: New Cyclin K Degraders from Old CDK Inhibitors. ACS chemical biology 19 (1) (2024)
Katie L Thomas, Habib Bouguenina, Daniel S J Miller, Fernando J Sialana, Thomas G Hayhow, Jyoti S Choudhary, Olivia W Rossanese, Benjamin R Bellenie
Degradation by Design: New Cyclin K Degraders from Old CDK Inhibitors. ACS chemical biology 19 (1) (2024)
Katie L Thomas, Habib Bouguenina, Daniel S J Miller, Fernando J Sialana, Thomas G Hayhow, Jyoti S Choudhary, Olivia W Rossanese, Benjamin R Bellenie
Degradation by Design: New Cyclin K Degraders from Old CDK Inhibitors. ACS chemical biology 19 (1) (2024)
Katie L Thomas, Habib Bouguenina, Daniel S J Miller, Fernando J Sialana, Thomas G Hayhow, Jyoti S Choudhary, Olivia W Rossanese, Benjamin R Bellenie
Degradation by Design: New Cyclin K Degraders from Old CDK Inhibitors. ACS chemical biology 19 (1) (2024)
Alice C Harnden, Owen A Davis, Gary M Box, Angela Hayes, Louise D Johnson, Alan T Henley, Alexis K de Haven Brandon, Melanie Valenti, Kwai-Ming J Cheung, Alfie Brennan, Rosemary Huckvale, Olivier A Pierrat, Rachel Talbot, Michael D Bright, Hafize Aysin Akpinar, Daniel S J Miller, Dalia Tarantino, Sharon Gowan, Selby de Klerk, Peter Craig McAndrew, Yann-Vaï Le Bihan, Mirco Meniconi, Rosemary Burke, Vladimir Kirkin, Rob L M van Montfort, Florence I Raynaud, Olivia W Rossanese, Benjamin R Bellenie, Swen Hoelder
Discovery of an In Vivo Chemical Probe for BCL6 Inhibition by Optimization of Tricyclic Quinolinones. Journal of medicinal chemistry (2023)
Manjuan Liu, Amin Mirza, Peter Craig McAndrew, Arjun Thapaliya, Olivier A Pierrat, Mark Stubbs, Tamas Hahner, Nicola E A Chessum, Paolo Innocenti, John Caldwell, Matthew D Cheeseman, Benjamin R Bellenie, Rob L M van Montfort, Gary K Newton, Rosemary Burke, Ian Collins, Swen Hoelder
Determination of Ligand-Binding Affinity ( K d ) Using Transverse Relaxation Rate ( R 2 ) in the Ligand-Observed 1 H NMR Experiment and Applications to Fragment-Based Drug Discovery. Journal of medicinal chemistry (2023)
Owen A Davis, Kwai-Ming J Cheung, Alfie Brennan, Matthew G Lloyd, Matthew J Rodrigues, Olivier A Pierrat, Gavin W Collie, Yann-Vaï Le Bihan, Rosemary Huckvale, Alice C Harnden, Ana Varela, Michael D Bright, Paul Eve, Angela Hayes, Alan T Henley, Michael D Carter, P Craig McAndrew, Rachel Talbot, Rosemary Burke, Rob L M van Montfort, Florence I Raynaud, Olivia W Rossanese, Mirco Meniconi, Benjamin R Bellenie, Swen Hoelder
Optimizing Shape Complementarity Enables the Discovery of Potent Tricyclic BCL6 Inhibitors. Journal of medicinal chemistry 65 (12) (2022)
Rosemary Huckvale, Alice C Harnden, Kwai-Ming J Cheung, Olivier A Pierrat, Rachel Talbot, Gary M Box, Alan T Henley, Alexis K de Haven Brandon, Albert E Hallsworth, Michael D Bright, Hafize Aysin Akpinar, Daniel S J Miller, Dalia Tarantino, Sharon Gowan, Angela Hayes, Emma A Gunnell, Alfie Brennan, Owen A Davis, Louise D Johnson, Selby de Klerk, Craig McAndrew, Yann-Vaï Le Bihan, Mirco Meniconi, Rosemary Burke, Vladimir Kirkin, Rob L M van Montfort, Florence I Raynaud, Olivia W Rossanese, Benjamin R Bellenie, Swen Hoelder
Improved Binding Affinity and Pharmacokinetics Enable Sustained Degradation of BCL6 In Vivo . Journal of medicinal chemistry 65 (12) (2022)
Matthew G Lloyd, Rosemary Huckvale, Kwai-Ming J Cheung, Matthew J Rodrigues, Gavin W Collie, Olivier A Pierrat, Mahad Gatti Iou, Michael Carter, Owen A Davis, P Craig McAndrew, Emma Gunnell, Yann-Vaï Le Bihan, Rachel Talbot, Alan T Henley, Louise D Johnson, Angela Hayes, Michael D Bright, Florence I Raynaud, Mirco Meniconi, Rosemary Burke, Rob L M van Montfort, Olivia W Rossanese, Benjamin R Bellenie, Swen Hoelder
Into Deep Water: Optimizing BCL6 Inhibitors by Growing into a Solvated Pocket. Journal of medicinal chemistry 64 (23) (2021)
Benjamin R Bellenie, Edward Hall, Ian Bruce, Matthew Spendiff, Andrew Culshaw, Sarah McDonald, Ameet Ambarkhane, Colin Chinn, Matthew Thomas, Elisabeth Rosner, Marguerite Bracher, Paul Nicklin, Stephen Marshall, Julie Coote, Eva Cullen, Clemence Tessier, Kuno Wuersch, Ajay Lal, Gillian Wallis, Gregory J Hollingworth, James Neef
Discovery and Toxicological Profiling of Aminopyridines as Orally Bioavailable Selective Inhibitors of PI3-Kinase γ. Journal of medicinal chemistry 64 (16) (2021)
Benjamin R Bellenie, Kwai-Ming J Cheung, Ana Varela, Olivier A Pierrat, Gavin W Collie, Gary M Box, Michael D Bright, Sharon Gowan, Angela Hayes, Matthew J Rodrigues, Kartika N Shetty, Michael Carter, Owen A Davis, Alan T Henley, Paolo Innocenti, Louise D Johnson, Manjuan Liu, Selby de Klerk, Yann-Vaï Le Bihan, Matthew G Lloyd, P Craig McAndrew, Erald Shehu, Rachel Talbot, Hannah L Woodward, Rosemary Burke, Vladimir Kirkin, Rob L M van Montfort, Florence I Raynaud, Olivia W Rossanese, Swen Hoelder
Achieving In Vivo Target Depletion through the Discovery and Optimization of Benzimidazolone BCL6 Degraders. Journal of medicinal chemistry 63 (8) (2020)

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Publication Activity (10 Years)

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Benjamin R Bellenie