Luca Gentilucci

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 23

Top Topics

Emergency Department

Molecular Docking

Top Venues

Molecules (Basel, Switzerland)

Journal of medicinal chemistry

International journal of molecular sciences

This page only lists publications with an associated author ORCID identifier.

Publications

Tingting He, Daria Giacomini, Alessandra Tolomelli, Monica Baiula, Luca Gentilucci
Conjecturing about Small-Molecule Agonists and Antagonists of α4β1 Integrin: From Mechanistic Insight to Potential Therapeutic Applications. Biomedicines 12 (2) (2024)
Tingting He, Daria Giacomini, Alessandra Tolomelli, Monica Baiula, Luca Gentilucci
Conjecturing about Small-Molecule Agonists and Antagonists of α4β1 Integrin: From Mechanistic Insight to Potential Therapeutic Applications. Biomedicines 12 (2) (2024)
Federica Santino, Luca Gentilucci
Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects. Molecules (Basel, Switzerland) 28 (1) (2023)
Michele Anselmi, Monica Baiula, Santi Spampinato, Roberto Artali, Tingting He, Luca Gentilucci
Design and Pharmacological Characterization of α 4 β 1 Integrin Cyclopeptide Agonists: Computational Investigation of Ligand Determinants for Agonism versus Antagonism. Journal of medicinal chemistry (2023)
Federica Santino, Luca Gentilucci
Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects. Molecules (Basel, Switzerland) 28 (1) (2023)
Federica Santino, Luca Gentilucci
Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects. Molecules (Basel, Switzerland) 28 (1) (2023)
Monica Baiula, Michele Anselmi, Francesco Musiani, Alessia Ghidini, Jacopo Carbone, Alberto Caligiana, Andrea Maurizio, Santi Spampinato, Luca Gentilucci
Design, Pharmacological Characterization, and Molecular Docking of Minimalist Peptidomimetic Antagonists of α 4 β 1 Integrin. International journal of molecular sciences 24 (11) (2023)
Junwei Zhao, Jacopo Carbone, Giovanna Farruggia, Anna Janecka, Luca Gentilucci, Natalia Calonghi
Synthesis and Antiproliferative Activity against Cancer Cells of Indole-Aryl-Amide Derivatives. Molecules (Basel, Switzerland) 28 (1) (2022)
Junwei Zhao, Jacopo Carbone, Giovanna Farruggia, Anna Janecka, Luca Gentilucci, Natalia Calonghi
Synthesis and Antiproliferative Activity against Cancer Cells of Indole-Aryl-Amide Derivatives. Molecules (Basel, Switzerland) 28 (1) (2022)
Jacopo Carbone, Alessia Ghidini, Antonio Romano, Luca Gentilucci, Francesco Musiani
PacDOCK: A Web Server for Positional Distance-Based and Interaction-Based Analysis of Docking Results. Molecules (Basel, Switzerland) 27 (20) (2022)
Junwei Zhao, Jacopo Carbone, Giovanna Farruggia, Anna Janecka, Luca Gentilucci, Natalia Calonghi
Synthesis and Antiproliferative Activity against Cancer Cells of Indole-Aryl-Amide Derivatives. Molecules (Basel, Switzerland) 28 (1) (2022)
Karol Wtorek, Alessia Ghidini, Luca Gentilucci, Anna Adamska-Bartłomiejczyk, Justyna Piekielna-Ciesielska, Chiara Ruzza, Chiara Sturaro, Girolamo Calò, Stefano Pieretti, Alicja Kluczyk, John McDonald, David G Lambert, Anna Janecka
Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors. International journal of molecular sciences 23 (20) (2022)
Michele Anselmi, Monica Baiula, Federica Santino, Junwei Zhao, Santi Spampinato, Natalia Calonghi, Luca Gentilucci
Design of α/β-Hybrid Peptide Ligands of α4β1 Integrin Equipped with a Linkable Side Chain for Chemoselective Biofunctionalization of Microstructured Materials. Biomedicines 9 (11) (2021)
Michele Anselmi, Pasquale Stavole, Elisa Boanini, Adriana Bigi, Eusebio Juaristi, Luca Gentilucci
Green synthesis of bioactive oligopeptides promoted by recyclable nanocrystalline hydroxyapatite. Future medicinal chemistry 12 (6) (2020)
Justyna Piekielna-Ciesielska, Roberto Artali, Ammar A H Azzam, David G Lambert, Alicja Kluczyk, Luca Gentilucci, Anna Janecka
Pharmacological Characterization of µ-Opioid Receptor Agonists with Biased G Protein or β-Arrestin Signaling, and Computational Study of Conformational Changes during Receptor Activation. Molecules (Basel, Switzerland) 26 (1) (2020)
Rossella De Marco, Enrico Rampazzo, Junwei Zhao, Luca Prodi, Mayra Paolillo, Pierre Picchetti, Francesca Gallo, Natalia Calonghi, Luca Gentilucci
Integrin-Targeting Dye-Doped PEG-Shell/Silica-Core Nanoparticles Mimicking the Proapoptotic Smac/DIABLO Protein. Nanomaterials (Basel, Switzerland) 10 (6) (2020)
Junwei Zhao, Federica Santino, Daria Giacomini, Luca Gentilucci
Integrin-Targeting Peptides for the Design of Functional Cell-Responsive Biomaterials. Biomedicines 8 (9) (2020)
Michele Anselmi, Adina Borbély, Eduard Figueras, Carmela Michalek, Isabell Kemker, Luca Gentilucci, Norbert Sewald
Linker Hydrophilicity Modulates the Anticancer Activity of RGD-Cryptophycin Conjugates. Chemistry (Weinheim an der Bergstrasse, Germany) 27 (3) (2020)
Giulia Martelli, Monica Baiula, Alberto Caligiana, Paola Galletti, Luca Gentilucci, Roberto Artali, Santi Spampinato, Daria Giacomini
Could Dissecting the Molecular Framework of β-Lactam Integrin Ligands Enhance Selectivity? Journal of medicinal chemistry 62 (22) (2019)
Rossella De Marco, Junwei Zhao, Arianna Greco, Simone Ioannone, Luca Gentilucci
In-Peptide Synthesis of Imidazolidin-2-one Scaffolds, Equippable with Proteinogenic or Taggable/Linkable Side Chains, General Promoters of Unusual Secondary Structures. The Journal of organic chemistry 84 (9) (2019)
Rossella De Marco, Andrea Bedini, Santi Spampinato, Lorenzo Comellini, Junwei Zhao, Roberto Artali, Luca Gentilucci
Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist. Journal of medicinal chemistry 61 (13) (2018)
Samantha Deianira Dattoli, Monica Baiula, Rossella De Marco, Andrea Bedini, Michele Anselmi, Luca Gentilucci, Santi Spampinato
DS-70, a novel and potent α4 integrin antagonist, is an effective treatment for experimental allergic conjunctivitis in guinea pigs. British journal of pharmacology 175 (20) (2018)
Rossella De Marco, Arianna Greco, Natalia Calonghi, Samantha D Dattoli, Monica Baiula, Santi Spampinato, Pierre Picchetti, Luisa De Cola, Michele Anselmi, Francesca Cipriani, Luca Gentilucci
Selective detection of α4β1 integrin (VLA-4)-expressing cells using peptide-functionalized nanostructured materials mimicking endothelial surfaces adjacent to inflammatory sites. Biopolymers (2017)