Stephan Rigol

Publication Activity (10 Years)

Years Active: 2017-2022
Publications (10 Years): 12

Top Topics

Metastatic Breast Cancer

Drug Administration

Molecular Docking

Acinetobacter Baumannii

Top Venues

Journal of the American Chemical Society

The Journal of organic chemistry

Proceedings of the National Academy of Sciences of the United States of America

Accounts of chemical research

This page only lists publications with an associated author ORCID identifier.

Publications

Kyriacos C Nicolaou, Saiyong Pan, Yogesh Shelke, Stephan Rigol, Ruiyang Bao, Dipendu Das, Qiuji Ye
A unified strategy for the total syntheses of eribulin and a macrolactam analogue of halichondrin B. Proceedings of the National Academy of Sciences of the United States of America 119 (32) (2022)
Kyriacos C Nicolaou, Saiyong Pan, Kiran K Pulukuri, Qiuji Ye, Stephan Rigol, Rohan D Erande, Dionisios Vourloumis, Bogusław P Nocek, Stefan Munneke, Joseph Lyssikatos, Amanda Valdiosera, Christine Gu, Baiwei Lin, Hetal Sarvaiaya, Jose Trinidad, Joseph Sandoval, Christina Lee, Mikhail Hammond, Monette Aujay, Nicole Taylor, Marybeth Pysz, James W Purcell, Julia Gavrilyuk
Design, Synthesis, and Biological Evaluation of Tubulysin Analogues, Linker-Drugs, and Antibody-Drug Conjugates, Insights into Structure-Activity Relationships, and Tubulysin-Tubulin Binding Derived from X-ray Crystallographic Analysis. The Journal of organic chemistry 86 (4) (2021)
Kyriacos C Nicolaou, Saiyong Pan, Yogesh Shelke, Qiuji Ye, Dipendu Das, Stephan Rigol
A Highly Convergent Total Synthesis of Norhalichondrin B. Journal of the American Chemical Society (2021)
Kyriacos C Nicolaou, Saiyong Pan, Yogesh G Shelke, Dipendu Das, Qiuji Ye, Yong Lu, Susanta Sau, Ruiyang Bao, Stephan Rigol
A Reverse Approach to the Total Synthesis of Halichondrin B. Journal of the American Chemical Society 143 (24) (2021)
Kyriacos C Nicolaou, Stephan Rigol, Emmanuel N Pitsinos, Dipendu Das, Yong Lu, Subhrajit Rout, Alexander W Schammel, Dane Holte, Baiwei Lin, Christine Gu, Hetal Sarvaiya, Jose Trinidad, Nicole Barbour, Amanda M Valdiosera, Joseph Sandoval, Christina Lee, Monette Aujay, Hanan Fernando, Anukriti Dhar, Holger Karsunky, Nicole Taylor, Marybeth Pysz, Julia Gavrilyuk
Uncialamycin-based antibody-drug conjugates: Unique enediyne ADCs exhibiting bystander killing effect. Proceedings of the National Academy of Sciences of the United States of America 118 (25) (2021)
Kyriacos C Nicolaou, Stephan Rigol
The Role of Organic Synthesis in the Emergence and Development of Antibody-Drug Conjugates as Targeted Cancer Therapies. Angewandte Chemie (International ed. in English) 58 (33) (2019)
Kyriacos C Nicolaou, Kiran Kumar Pulukuri, Stephan Rigol, Zisis Peitsinis, Ruocheng Yu, Satoshi Kishigami, Nicholas Cen, Monette Aujay, Joseph Sandoval, Nancy Zepeda, Julia Gavrilyuk
Correction to "Short Total Synthesis of Δ12-Prostaglandin J2 and Related Prostaglandins. Design, Synthesis, and Biological Evaluation of Macrocyclic Δ12-Prostaglandin J2 Analogues". The Journal of organic chemistry 84 (4) (2019)
Kyriacos C Nicolaou, Kiran Kumar Pulukuri, Stephan Rigol, Zisis Peitsinis, Ruocheng Yu, Satoshi Kishigami, Nicholas Cen, Monette Aujay, Joseph Sandoval, Nancy Zepeda, Julia Gavrilyuk
Short Total Synthesis of Δ12-Prostaglandin J2 and Related Prostaglandins. Design, Synthesis, and Biological Evaluation of Macrocyclic Δ12-Prostaglandin J2 Analogues. The Journal of organic chemistry 84 (1) (2018)
Kyriacos C Nicolaou, Stephan Rigol
Total Synthesis in Search of Potent Antibody-Drug Conjugate Payloads. From the Fundamentals to the Translational. Accounts of chemical research 52 (1) (2018)
Kyriacos C Nicolaou, Kiran Kumar Pulukuri, Stephan Rigol, Marek Buchman, Akshay A Shah, Nicholas Cen, Megan D McCurry, Kathryn Beabout, Yousif Shamoo
Enantioselective Total Synthesis of Antibiotic CJ-16,264, Synthesis and Biological Evaluation of Designed Analogues, and Discovery of Highly Potent and Simpler Antibacterial Agents. Journal of the American Chemical Society 139 (44) (2017)
Kathryn Beabout, Megan D McCurry, Heer Mehta, Akshay A Shah, Kiran Kumar Pulukuri, Stephan Rigol, Yanping Wang, Kyriacos C Nicolaou, Yousif Shamoo
Experimental Evolution of Diverse Strains as a Method for the Determination of Biochemical Mechanisms of Action for Novel Pyrrolizidinone Antibiotics. ACS infectious diseases 3 (11) (2017)
Kyriacos C Nicolaou, Pengxi Chen, Shugao Zhu, Quan Cai, Rohan D Erande, Ruofan Li, Hongbao Sun, Kiran Kumar Pulukuri, Stephan Rigol, Monette Aujay, Joseph Sandoval, Julia Gavrilyuk
Streamlined Total Synthesis of Trioxacarcins and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues Thereof. Discovery of Simpler Designed and Potent Trioxacarcin Analogues. Journal of the American Chemical Society 139 (43) (2017)