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Experimental and new investigational drugs for the treatment of uterine fibroids.

Giulio EvangelistiSimone FerreroUmberto PerroneClaudio GustavinoEugenio VolpiAlberto IzzottiFabio Barra
Published in: Expert opinion on investigational drugs (2024)
Despite ulipristal acetate's well-established efficacy as a selective progesterone receptor modulator (SPRM) in fibroid treatment, its prescription has declined due to the rare but severe risk of liver damage. Oral GnRH antagonists, like elagolix, relugolix, and linzagolix, with their novel pharmacodynamic properties, are gaining traction in fibroid management, inducing a dose-dependent reduction in circulating sex hormone levels. Ongoing research on natural compounds, such as vitamin D and epigallocatechin gallate (EGCG), presents emerging options for treating uterine fibroids. This evolving landscape reflects the ongoing efforts to improve therapeutic outcomes for individuals with symptomatic uterine fibroids.
Keyphrases
  • randomized controlled trial
  • early onset
  • pregnancy outcomes
  • clinical trial
  • combination therapy
  • single cell
  • pregnant women
  • study protocol
  • open label
  • phase ii
  • weight loss
  • double blind