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Olutasidenib (FT-2102) in patients with relapsed or refractory IDH1-mutant glioma: a multicenter, open-label, phase 1b/2 trial.

Macarena I de la FuenteHoward ColmanMark RosenthalBrian A Van TineDanijela LevacicTobias WalbertHui K GanMaria VieitoMohammed M MilhemKathryn LipfordSanjeev ForsythSylvie M GuichardYelena MikhailovAlexander SedkovJulie BrevardPatrick F KellyHesham MohamedVarun Monga
Published in: Neuro-oncology (2022)
Olutasidenib 150 mg BID was well tolerated in patients with relapsed/refractory gliomas harboring an IDH1  R132X mutation and demonstrated preliminary evidence of clinical activity in this heavily pretreated population.
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