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p-Cymene Complexes of Ruthenium(II) as Antitumor Agents.

María Angeles Pujante-GaliánSergio A PérezMercedes G MontalbánGuzmán CarissimiMarta G FusterGloria VílloraGabriel García
Published in: Molecules (Basel, Switzerland) (2020)
In this work, the cytotoxic behavior of six ruthenium(II) complexes of stoichiometry [(η6-p-cymene)RuCl2L] (I-VI), L = 4-cyanopyridine (I), 2-aminophenol (II), 4-aminophenol (III), pyridazine (IV), and [(η6-p-cymene)RuClL2]PF6; L = cyanopyridine (V), L = 2-aminophenol(VI) towards three cell lines was studied. Two of them, HeLa and MCF-7, are human carcinogenic cells from cervical carcinoma and human breast cancer, respectively. A comparison with healthy cells was carried out with BGM cells which are monkey epithelial cells of renal origin. The behavior of complex II exhibits selectivity towards healthy cells, which is a promising feature for use in cancer treatment since it might reduce the side effects of most current therapies.
Keyphrases
  • induced apoptosis
  • cell cycle arrest
  • endothelial cells
  • endoplasmic reticulum stress
  • machine learning
  • signaling pathway
  • deep learning
  • induced pluripotent stem cells
  • cell proliferation
  • pluripotent stem cells