Clinically relevant CHK1 inhibitors abrogate wild-type and Y537S mutant ERα expression and proliferation in luminal primary and metastatic breast cancer cells.
Sara PescatoriStefano LeoneManuela CipollettiStefania BartoloniAlessandra di MasiFilippo AcconciaPublished in: Journal of experimental & clinical cancer research : CR (2022)
CHK1 could be considered as an appealing novel pharmacological target for the treatment of luminal primary and MBCs.