Arthur E Jacobson

Publication Activity (10 Years)

Years Active: 2020-2024
Publications (10 Years): 17

Top Topics

Molecular Docking

Structure Activity Relationship

Capillary Electrophoresis

Pain Management

Top Venues

Molecules (Basel, Switzerland)

RSC medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Hudson G Roth, Madhurima Das, Agnieszka Sulima, Dan Luo, Sophia Kaska, Thomas Edward Prisinzano, Andrew T Kerr, Arthur E Jacobson, Kenner C Rice
Functional Activity of Enantiomeric Oximes and Diastereomeric Amines and Cyano Substituents at C9 in 3-Hydroxy- N -phenethyl-5-phenylmorphans. Molecules (Basel, Switzerland) 29 (9) (2024)
Hudson G Roth, Madhurima Das, Agnieszka Sulima, Dan Luo, Sophia Kaska, Thomas Edward Prisinzano, Andrew T Kerr, Arthur E Jacobson, Kenner C Rice
Functional Activity of Enantiomeric Oximes and Diastereomeric Amines and Cyano Substituents at C9 in 3-Hydroxy- N -phenethyl-5-phenylmorphans. Molecules (Basel, Switzerland) 29 (9) (2024)
Joshua A Lutz, Agnieszka Sulima, Eugene S Gutman, Eric W Bow, Dan Luo, Sophia Kaska, Thomas Edward Prisinzano, Carol A Paronis, Jack Bergman, Gregory H Imler, Andrew T Kerr, Arthur E Jacobson, Kenner C Rice
Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans. Molecules (Basel, Switzerland) 28 (12) (2023)
Dana R Chambers, Agnieszka Sulima, Dan Luo, Thomas Edward Prisinzano, Arthur E Jacobson, Kenner C Rice
A MOR Antagonist with High Potency and Antagonist Efficacy among Diastereomeric C9-Alkyl-Substituted N -Phenethyl-5-(3-hydroxy)phenylmorphans. Molecules (Basel, Switzerland) 28 (14) (2023)
Joshua A Lutz, Agnieszka Sulima, Eugene S Gutman, Eric W Bow, Dan Luo, Sophia Kaska, Thomas Edward Prisinzano, Carol A Paronis, Jack Bergman, Gregory H Imler, Andrew T Kerr, Arthur E Jacobson, Kenner C Rice
Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans. Molecules (Basel, Switzerland) 28 (12) (2023)
Joshua A Lutz, Agnieszka Sulima, Eugene S Gutman, Eric W Bow, Dan Luo, Sophia Kaska, Thomas Edward Prisinzano, Carol A Paronis, Jack Bergman, Gregory H Imler, Andrew T Kerr, Arthur E Jacobson, Kenner C Rice
Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans. Molecules (Basel, Switzerland) 28 (12) (2023)
Madhurima Das, George W Ward, Agnieszka Sulima, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Andrew T Kerr, Arthur E Jacobson, Kenner C Rice
Potent MOR Agonists from 2'-Hydroxy-5,9-dimethyl- N -phenethyl Substituted-6,7-benzomorphans and from C8-Hydroxy, Methylene and Methyl Derivatives of N -Phenethylnormetazocine. Molecules (Basel, Switzerland) 28 (23) (2023)
Fuying Li, Theresa A Kopajtic, Jonathan L Katz, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans. Molecules (Basel, Switzerland) 27 (24) (2022)
Fuying Li, Theresa A Kopajtic, Jonathan L Katz, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans. Molecules (Basel, Switzerland) 27 (24) (2022)
Fuying Li, Theresa A Kopajtic, Jonathan L Katz, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans. Molecules (Basel, Switzerland) 27 (24) (2022)
Fuying Li, Theresa A Kopajtic, Jonathan L Katz, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans. Molecules (Basel, Switzerland) 27 (24) (2022)
Fuying Li, Theresa A Kopajtic, Jonathan L Katz, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans. Molecules (Basel, Switzerland) 27 (24) (2022)
Dana R Chambers, Agnieszka Sulima, Dan Luo, Thomas Edward Prisinzano, Alexander Goldberg, Bing Xie, Lei Shi, Carol A Paronis, Jack Bergman, Nima Nassehi, Dana E Selley, Gregory H Imler, Arthur E Jacobson, Kenner C Rice
A Journey through Diastereomeric Space: The Design, Synthesis, In Vitro and In Vivo Pharmacological Activity, and Molecular Modeling of Novel Potent Diastereomeric MOR Agonists and Antagonists. Molecules (Basel, Switzerland) 27 (19) (2022)
Fuying Li, Theresa A Kopajtic, Jonathan L Katz, Dan Luo, Thomas Edward Prisinzano, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans. Molecules (Basel, Switzerland) 27 (24) (2022)
Agnieszka Sulima, Fuying Li, Jeffrey Brian Morgan, Phong Truong, Joshua F G Antoline, Therese Oertel, Rodell C Barrientos, Oscar B Torres, Zoltan Beck, Gregory H Imler, Jeffrey R Deschamps, Gary R Matyas, Arthur E Jacobson, Kenner C Rice
Design, Synthesis, and In Vivo Evaluation of C1-Linked 4,5-Epoxymorphinan Haptens for Heroin Vaccines. Molecules (Basel, Switzerland) 27 (5) (2022)
Essie Komla, Oscar B Torres, Rashmi Jalah, Agnieszka Sulima, Zoltan Beck, Carl R Alving, Arthur E Jacobson, Kenner C Rice, Gary R Matyas
Effect of Preexisting Immunity to Tetanus Toxoid on the Efficacy of Tetanus Toxoid-Conjugated Heroin Vaccine in Mice. Vaccines 9 (6) (2021)
Eugene S Gutman, Eric Bow, Fuying Li, Agnieszka Sulima, Sophia Kaska, Rachel Crowley, Thomas Edward Prisinzano, Yong-Sok Lee, Sergio A Hassan, Gregory H Imler, Jeffrey R Deschamps, Arthur E Jacobson, Kenner C Rice
G-Protein biased opioid agonists: 3-hydroxy-N-phenethyl-5-phenylmorphans with three-carbon chain substituents at C9. RSC medicinal chemistry 11 (8) (2020)