Atsushi Kittaka

Publication Activity (10 Years)

Years Active: 2019-2024
Publications (10 Years): 18

Top Topics

Acute Myeloid Leukemia

Molecular Docking

Binding Protein

Top Venues

International journal of molecular sciences

ACS chemical biology

The Journal of organic chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Carole Peluso-Iltis, Noé Pierrat, Daniela Rovito, Judit Osz, Daisuke Sawada, Atsushi Kittaka, Gilles Laverny, Natacha Rochel
4-Hydroxy-1α,25-Dihydroxyvitamin D 3 : Synthesis and Structure-Function Study. Biomolecules 14 (5) (2024)
Michiyasu Ishizawa, Masashi Takano, Atsushi Kittaka, Taro Matsumoto, Makoto Makishima
2α-Substituted Vitamin D Derivatives Effectively Enhance the Osteoblast Differentiation of Dedifferentiated Fat Cells. Biomolecules 14 (6) (2024)
Michiyasu Ishizawa, Masashi Takano, Atsushi Kittaka, Taro Matsumoto, Makoto Makishima
2α-Substituted Vitamin D Derivatives Effectively Enhance the Osteoblast Differentiation of Dedifferentiated Fat Cells. Biomolecules 14 (6) (2024)
Carole Peluso-Iltis, Noé Pierrat, Daniela Rovito, Judit Osz, Daisuke Sawada, Atsushi Kittaka, Gilles Laverny, Natacha Rochel
4-Hydroxy-1α,25-Dihydroxyvitamin D 3 : Synthesis and Structure-Function Study. Biomolecules 14 (5) (2024)
Fumihiro Kawagoe, Sayuri Mototani, Atsushi Kittaka
Efficient Stereo-Selective Fluorination on Vitamin D 3 Side-Chain Using Electrophilic Fluorination. Biomolecules 14 (1) (2023)
Fumihiro Kawagoe, Sayuri Mototani, Atsushi Kittaka
Efficient Stereo-Selective Fluorination on Vitamin D 3 Side-Chain Using Electrophilic Fluorination. Biomolecules 14 (1) (2023)
Fumihiro Kawagoe, Sayuri Mototani, Atsushi Kittaka
Efficient Stereo-Selective Fluorination on Vitamin D 3 Side-Chain Using Electrophilic Fluorination. Biomolecules 14 (1) (2023)
Fumihiro Kawagoe, Sayuri Mototani, Aileen Mendoza, Yasushi Takemoto, Motonari Uesugi, Atsushi Kittaka
Structure-activity relationship studies on vitamin D-based selective SREBP/SCAP inhibitor KK-052. RSC medicinal chemistry 14 (10) (2023)
Fumihiro Kawagoe, Sayuri Mototani, Kaori Yasuda, Akiko Takeuchi, Hiroki Mano, Shinji Kakuda, Hiroshi Saitoh, Toshiyuki Sakaki, Atsushi Kittaka
Synthesis of (22 R )-, (22 S )-22-Fluoro-, and 22,22-Difluoro-25-hydroxyvitamin D 3 and Effects of Side-Chain Fluorination on Biological Activity and CYP24A1-Dependent Metabolism. The Journal of organic chemistry (2023)
Yuka Mizumoto, Ryota Sakamoto, Akiko Nagata, Suzuka Sakane, Atsushi Kittaka, Minami Odagi, Masayuki Tera, Kazuo Nagasawa
Synthesis of C2-Alkoxy-Substituted 19-Nor Vitamin D 3 Derivatives: Stereoselectivity and Biological Activity. Biomolecules 12 (1) (2022)
Sayuri Mototani, Fumihiro Kawagoe, Kaori Yasuda, Hiroki Mano, Toshiyuki Sakaki, Atsushi Kittaka
The First Convergent Synthesis of 23,23-Difluoro-25-hydroxyvitamin D 3 and Its 24-Hydroxy Derivatives: Preliminary Assessment of Biological Activities. Molecules (Basel, Switzerland) 27 (16) (2022)
Fumihiro Kawagoe, Aileen Mendoza, Yuki Hayata, Lisa Asano, Kenjiro Kotake, Sayuri Mototani, Satoshi Kawamura, Shigeyuki Kurosaki, Yusuke Akagi, Yasushi Takemoto, Kazuo Nagasawa, Hayato Nakagawa, Motonari Uesugi, Atsushi Kittaka
Discovery of a Vitamin D Receptor-Silent Vitamin D Derivative That Impairs Sterol Regulatory Element-Binding Protein In Vivo. Journal of medicinal chemistry 64 (9) (2021)
Kaori Yasuda, Miyu Nishikawa, Hiroki Mano, Masashi Takano, Atsushi Kittaka, Shinichi Ikushiro, Toshiyuki Sakaki
Development of In Vitro and In Vivo Evaluation Systems for Vitamin D Derivatives and Their Application to Drug Discovery. International journal of molecular sciences 22 (21) (2021)
Fumihiro Kawagoe, Sayuri Mototani, Atsushi Kittaka
The Synthesis and Biological Evaluation of D-Ring-Modified Vitamin D Analogues. Biomolecules 11 (11) (2021)
Fumihiro Kawagoe, Sayuri Mototani, Kaori Yasuda, Hiroki Mano, Toshiyuki Sakaki, Atsushi Kittaka
Stereoselective Synthesis of 24-Fluoro-25-Hydroxyvitamin D3 Analogues and Their Stability to hCYP24A1-Dependent Catabolism. International journal of molecular sciences 22 (21) (2021)
Fumihiro Kawagoe, Sayuri Mototani, Atsushi Kittaka
Design and Synthesis of Fluoro Analogues of Vitamin D. International journal of molecular sciences 22 (15) (2021)
Daisuke Sawada, Shinji Kakuda, Akiko Takeuchi, Fumihiro Kawagoe, Midori Takimoto-Kamimura, Atsushi Kittaka
Effects of 2-substitution on 14-epi-19-nortachysterol-mediated biological events: based on synthesis and X-ray co-crystallographic analysis with the human vitamin D receptor. Organic & biomolecular chemistry 16 (14) (2019)
Akiko Nagata, Yusuke Akagi, Lisa Asano, Kenjiro Kotake, Fumihiro Kawagoe, Aileen Mendoza, Shadi Sedghi Masoud, Kosuke Usuda, Koji Yasui, Yasushi Takemoto, Atsushi Kittaka, Kazuo Nagasawa, Motonari Uesugi
Synthetic Chemical Probes That Dissect Vitamin D Activities. ACS chemical biology 14 (12) (2019)