Julian Blagg
Publication Activity (10 Years)
Years Active: 2016-2019
Publications (10 Years): 5
Publications (10 Years): 5
Publications
- Manjuan Liu, Aurélie Mallinger, Marcello Tortorici, Yvette Newbatt, Meirion Richards, Amin Mirza, Rob L M van Montfort, Rosemary Burke, Julian Blagg, Teresa Kaserer
- Hannah L Woodward, Paolo Innocenti, Kwai-Ming J Cheung, Angela Hayes, Jennie Roberts, Alan T Henley, Amir Faisal, Grace Wing-Yan Mak, Gary Box, Isaac M Westwood, Nora Cronin, Michael Carter, Melanie Valenti, Alexis De Haven Brandon, Lisa O'Fee, Harry Saville, Jessica Schmitt, Rosemary Burke, Fabio Broccatelli, Rob L M van Montfort, Florence I Raynaud, Suzanne A Eccles, Spiros Linardopoulos, Julian Blagg, Swen HoelderIntroduction of a Methyl Group Curbs Metabolism of Pyrido[3,4- d]pyrimidine Monopolar Spindle 1 (MPS1) Inhibitors and Enables the Discovery of the Phase 1 Clinical Candidate N2-(2-Ethoxy-4-(4-methyl-4 H-1,2,4-triazol-3-yl)phenyl)-6-methyl- N8-neopentylpyrido[3,4- d]pyrimidine-2,8-diamine (BOS172722). Journal of medicinal chemistry 61 (18) (2018)
- James A H Gilburt, Hajrah Sarkar, Peter Sheldrake, Julian Blagg, Liming Ying, Charlotte A Dodson
- Paul Andrew Clarke, Maria-Jesus Ortiz-Ruiz, Robert TePoele, Olajumoke Adeniji-Popoola, Gary Box, Will Court, Stephanie Czasch, Samer El Bawab, Christina Esdar, Ken Ewan, Sharon Gowan, Alexis De Haven Brandon, Phillip Hewitt, Stephen M Hobbs, Wolfgang Kaufmann, Aurélie Mallinger, Florence Raynaud, Toby Roe, Felix Rohdich, Kai Schiemann, Stephanie Simon, Richard Schneider, Melanie Valenti, Stefan Weigt, Julian Blagg, Andree Blaukat, Trevor C Dale, Suzanne A Eccles, Stefan Hecht, Klaus Urbahns, Paul Workman, Dirk Wienke