Samuele Cazzamalli

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 25

Top Topics

Human Serum Albumin

Top Venues

Journal of medicinal chemistry

Bioconjugate chemistry

Nature chemistry

European journal of nuclear medicine and molecular imaging

This page only lists publications with an associated author ORCID identifier.

Publications

Tony Georgiev, Lucrezia Principi, Andrea Galbiati, Ettore Gilardoni, Dario Neri, Samuele Cazzamalli
Targeted interleukin-2 enhances the in vivo anti-cancer activity of Pluvicto™. European journal of nuclear medicine and molecular imaging (2024)
Andrea Galbiati, Matilde Bocci, Silvia Gervasoni, Eleonora Prodi, Giuliano Malloci, Dario Neri, Samuele Cazzamalli
Molecular Evolution of Multivalent OncoFAP Derivatives with Enhanced Tumor Uptake and Prolonged Tumor Retention. Journal of medicinal chemistry (2024)
Andrea Galbiati, Matilde Bocci, Silvia Gervasoni, Eleonora Prodi, Giuliano Malloci, Dario Neri, Samuele Cazzamalli
Molecular Evolution of Multivalent OncoFAP Derivatives with Enhanced Tumor Uptake and Prolonged Tumor Retention. Journal of medicinal chemistry 67 (15) (2024)
Sara Puglioli, Mosè Fabbri, Claudia Comacchio, Laura Alvigini, Roberto De Luca, Sebastian Oehler, Ettore Gilardoni, Gabriele Bassi, Samuele Cazzamalli, Dario Neri, Nicholas Favalli
Permutational Encoding Strategy Accelerates HIT Validation from Single-Stranded DNA-Encoded Libraries. Bioconjugate chemistry 35 (7) (2024)
Marco Müller, Laura Lucaroni, Nicholas Favalli, Gabriele Bassi, Dario Neri, Samuele Cazzamalli, Sebastian Oehler
Discovery of Glutamate Carboxypeptidase III Ligands to Compete the Uptake of [ 177 Lu]Lu-PSMA-617 in Healthy Organs. Journal of medicinal chemistry 67 (10) (2024)
Giulia Rotta, Emanuele Puca, Samuele Cazzamalli, Dario Neri, Sheila Dakhel
Cytokine Biopharmaceuticals with "Activity-on-Demand" for Cancer Therapy. Bioconjugate chemistry 35 (8) (2024)
Sara Puglioli, Mosè Fabbri, Claudia Comacchio, Laura Alvigini, Roberto De Luca, Sebastian Oehler, Ettore Gilardoni, Gabriele Bassi, Samuele Cazzamalli, Dario Neri, Nicholas Favalli
Permutational Encoding Strategy Accelerates HIT Validation from Single-Stranded DNA-Encoded Libraries. Bioconjugate chemistry (2024)
Marco Müller, Laura Lucaroni, Nicholas Favalli, Gabriele Bassi, Dario Neri, Samuele Cazzamalli, Sebastian Oehler
Discovery of Glutamate Carboxypeptidase III Ligands to Compete the Uptake of [ 177 Lu]Lu-PSMA-617 in Healthy Organs. Journal of medicinal chemistry 67 (10) (2024)
Giulia Rotta, Emanuele Puca, Samuele Cazzamalli, Dario Neri, Sheila Dakhel
Cytokine Biopharmaceuticals with "Activity-on-Demand" for Cancer Therapy. Bioconjugate chemistry (2024)
Andrea Galbiati, Matilde Bocci, Silvia Gervasoni, Eleonora Prodi, Giuliano Malloci, Dario Neri, Samuele Cazzamalli
Molecular Evolution of Multivalent OncoFAP Derivatives with Enhanced Tumor Uptake and Prolonged Tumor Retention. Journal of medicinal chemistry 67 (15) (2024)
Tony Georgiev, Lucrezia Principi, Andrea Galbiati, Ettore Gilardoni, Dario Neri, Samuele Cazzamalli
Targeted interleukin-2 enhances the in vivo anti-cancer activity of Pluvicto™. European journal of nuclear medicine and molecular imaging 51 (8) (2024)
Marco Müller, Laura Lucaroni, Nicholas Favalli, Gabriele Bassi, Dario Neri, Samuele Cazzamalli, Sebastian Oehler
Discovery of Glutamate Carboxypeptidase III Ligands to Compete the Uptake of [ 177 Lu]Lu-PSMA-617 in Healthy Organs. Journal of medicinal chemistry (2024)
Aureliano Zana, Claudia Puig-Moreno, Matilde Bocci, Ettore Gilardoni, Cesare Di Nitto, Lucrezia Principi, Domenico Ravazza, Giulia Rotta, Eleonora Prodi, Roberto De Luca, Dario Neri, Samuele Cazzamalli
A Comparative Analysis of Fibroblast Activation Protein-Targeted Small Molecule-Drug, Antibody-Drug, and Peptide-Drug Conjugates. Bioconjugate chemistry (2023)
Sebastian Oehler, Laura Lucaroni, Francesca Migliorini, Abdullah Elsayed, Luca Prati, Sara Puglioli, Mattia Matasci, Kristina Schira, Jörg Scheuermann, Denis Yudin, Min Jia, Nenad Ban, David A Bushnell, Roger Kornberg, Samuele Cazzamalli, Dario Neri, Nicholas Favalli, Gabriele Bassi
A DNA-encoded chemical library based on chiral 4-amino-proline enables stereospecific isozyme-selective protein recognition. Nature chemistry (2023)
Wen Torng, Ilaria Biancofiore, Sebastian Oehler, Jin Xu, Jessica Xu, Ian Watson, Brenno Masina, Luca Prati, Nicholas Favalli, Gabriele Bassi, Dario Neri, Samuele Cazzamalli, Jianwen A Feng
Deep Learning Approach for the Discovery of Tumor-Targeting Small Organic Ligands from DNA-Encoded Chemical Libraries. ACS omega 8 (28) (2023)
Aureliano Zana, Andrea Galbiati, Ettore Gilardoni, Matilde Bocci, Jacopo Millul, Theo Sturm, Riccardo Stucchi, Abdullah Elsayed, Lisa Nadal, Martina Cirillo, Wolfgang Roll, Lars Stegger, Inga Asmus, Philipp Backhaus, Michael Schäfers, Dario Neri, Samuele Cazzamalli
Fibroblast Activation Protein triggers release of drug payload from non-internalizing small molecule-drug conjugates in solid tumors. Clinical cancer research : an official journal of the American Association for Cancer Research (2022)
Sheila Dakhel, Andrea Galbiati, Francesca Migliorini, Claudia Comacchio, Sebastian Oehler, Luca Prati, Jörg Scheuermann, Samuele Cazzamalli, Dario Neri, Gabriele Bassi, Nicholas Favalli
Isolation of a Natural Killer Group 2D Small-Molecule Ligand from DNA-Encoded Chemical Libraries. ChemMedChem 17 (21) (2022)
Nicholas Favalli, Gabriele Bassi, Christian Pellegrino, Jacopo Millul, Roberto De Luca, Samuele Cazzamalli, Su Yang, Anika Trenner, Nour L Mozaffari, Renier Myburgh, Mustafa Moroglu, Stuart J Conway, Alessandro A Sartori, Markus Gabriel Manz, Richard A Lerner, Peter K Vogt, Jörg Scheuermann, Dario Neri
Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications. Nature chemistry 13 (6) (2021)
Jacopo Millul, Gabriele Bassi, Jacqueline Mock, Abdullah Elsayed, Christian Pellegrino, Aureliano Zana, Sheila Dakhel Plaza, Lisa Nadal, Andreas Gloger, Eleonore Schmidt, Ilaria Biancofiore, Etienne J Donckele, Florent Samain, Dario Neri, Samuele Cazzamalli
An ultra-high-affinity small organic ligand of fibroblast activation protein for tumor-targeting applications. Proceedings of the National Academy of Sciences of the United States of America 118 (16) (2021)
Adrián Gironda-Martínez, Émile M D Gorre, Luca Prati, Jean-François Gosalbes, Sheila Dakhel, Samuele Cazzamalli, Florent Samain, Etienne J Donckele, Dario Neri
Identification and Validation of New Interleukin-2 Ligands Using DNA-Encoded Libraries. Journal of medicinal chemistry 64 (23) (2021)
Jacopo Millul, Christiane Krudewig, Aureliano Zana, Sheila Dakhel Plaza, Emanuele Puca, Alessandra Villa, Dario Neri, Samuele Cazzamalli
Immunotherapy with Immunocytokines and PD-1 Blockade Enhances the Anticancer Activity of Small Molecule-Drug Conjugates Targeting Carbonic Anhydrase IX. Molecular cancer therapeutics 20 (3) (2020)
Emanuele Puca, Philipp Probst, Marco Stringhini, Patrizia Murer, Giovanni Pellegrini, Samuele Cazzamalli, Cornelia Hutmacher, Baptiste Gouyou, Sarah Wulhfard, Mattia Matasci, Alessandra Villa, Dario Neri
The antibody-based delivery of interleukin-12 to solid tumors boosts NK and CD8+ T cell activity and synergizes with immune checkpoint inhibitors. International journal of cancer 146 (9) (2019)
Samuele Cazzamalli, Alberto Dal Corso, Fontaine Widmayer, Dario Neri
Chemically Defined Antibody- and Small Molecule-Drug Conjugates for in Vivo Tumor Targeting Applications: A Comparative Analysis. Journal of the American Chemical Society 140 (5) (2018)
Samuele Cazzamalli, Barbara Ziffels, Fontaine Widmayer, Patrizia Murer, Giovanni Pellegrini, Francesca Pretto, Sarah Wulhfard, Dario Neri
Enhanced Therapeutic Activity of Non-Internalizing Small-Molecule-Drug Conjugates Targeting Carbonic Anhydrase IX in Combination with Targeted Interleukin-2. Clinical cancer research : an official journal of the American Association for Cancer Research 24 (15) (2018)
Yizhou Li, Roberto De Luca, Samuele Cazzamalli, Francesca Pretto, Davor Bajic, Jörg Scheuermann, Dario Neri
Versatile protein recognition by the encoded display of multiple chemical elements on a constant macrocyclic scaffold. Nature chemistry 10 (4) (2018)