Stephen N Greszler (Stephen Greszler)

ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 18

Top Venues

Journal of medicinal chemistry

Organic letters

The Journal of organic chemistry

ACS omega

This page only lists publications with an associated author ORCID identifier.

Publications

Mathieu Pizzonero, Rhalid Akkari, Xavier Bock, Romain Gosmini, Elsa De Lemos, Béranger Duthion, Gregory Newsome, Thi-Thu-Trang Mai, Virginie Roques, Hélène Jary, Jean-Michel Lefrancois, Laetitia Cherel, Vanessa Quenehen, Marielle Babel, Nuria Merayo, Natacha Bienvenu, Oscar Mammoliti, Ghjuvanni Coti, Adeline Palisse, Marlon Cowart, Anurupa Shrestha, Stephen N Greszler, Steven Van Der Plas, Koen Jansen, Pieter Claes, Mia Jans, Maarten Gees, Monica Borgonovi, Gert De Wilde, Katja Conrath
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector. Journal of medicinal chemistry 67 (7) (2024)
Mathieu Pizzonero, Rhalid Akkari, Xavier Bock, Romain Gosmini, Elsa De Lemos, Béranger Duthion, Gregory Newsome, Thi-Thu-Trang Mai, Virginie Roques, Hélène Jary, Jean-Michel Lefrancois, Laetitia Cherel, Vanessa Quenehen, Marielle Babel, Nuria Merayo, Natacha Bienvenu, Oscar Mammoliti, Ghjuvanni Coti, Adeline Palisse, Marlon Cowart, Anurupa Shrestha, Stephen N Greszler, Steven Van Der Plas, Koen Jansen, Pieter Claes, Mia Jans, Maarten Gees, Monica Borgonovi, Gert De Wilde, Katja Conrath
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector. Journal of medicinal chemistry 67 (7) (2024)
Mathieu Pizzonero, Rhalid Akkari, Xavier Bock, Romain Gosmini, Elsa De Lemos, Béranger Duthion, Gregory Newsome, Thi-Thu-Trang Mai, Virginie Roques, Hélène Jary, Jean-Michel Lefrancois, Laetitia Cherel, Vanessa Quenehen, Marielle Babel, Nuria Merayo, Natacha Bienvenu, Oscar Mammoliti, Ghjuvanni Coti, Adeline Palisse, Marlon Cowart, Anurupa Shrestha, Stephen N Greszler, Steven Van Der Plas, Koen Jansen, Pieter Claes, Mia Jans, Maarten Gees, Monica Borgonovi, Gert De Wilde, Katja Conrath
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector. Journal of medicinal chemistry 67 (7) (2024)
Mathieu Pizzonero, Rhalid Akkari, Xavier Bock, Romain Gosmini, Elsa De Lemos, Béranger Duthion, Gregory Newsome, Thi-Thu-Trang Mai, Virginie Roques, Hélène Jary, Jean-Michel Lefrancois, Laetitia Cherel, Vanessa Quenehen, Marielle Babel, Nuria Merayo, Natacha Bienvenu, Oscar Mammoliti, Ghjuvanni Coti, Adeline Palisse, Marlon Cowart, Anurupa Shrestha, Stephen N Greszler, Steven Van Der Plas, Koen Jansen, Pieter Claes, Mia Jans, Maarten Gees, Monica Borgonovi, Gert De Wilde, Katja Conrath
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector. Journal of medicinal chemistry (2024)
Mathieu Pizzonero, Rhalid Akkari, Xavier Bock, Romain Gosmini, Elsa De Lemos, Béranger Duthion, Gregory Newsome, Thi-Thu-Trang Mai, Virginie Roques, Hélène Jary, Jean-Michel Lefrancois, Laetitia Cherel, Vanessa Quenehen, Marielle Babel, Nuria Merayo, Natacha Bienvenu, Oscar Mammoliti, Ghjuvanni Coti, Adeline Palisse, Marlon Cowart, Anurupa Shrestha, Stephen N Greszler, Steven Van Der Plas, Koen Jansen, Pieter Claes, Mia Jans, Maarten Gees, Monica Borgonovi, Gert De Wilde, Katja Conrath
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector. Journal of medicinal chemistry 67 (7) (2024)
Ashley L Ramos, Eric R Goedken, Kristine E Frank, Maria A Argiriadi, Sana Bazzaz, Zhiguo Bian, Jesse T C Brown, Paolo A Centrella, Hui-Ju Chen, Jeremy S Disch, Pamela L Donner, David B Duignan, Diana Gikunju, Stephen N Greszler, Marie-Aude Guié, Sevan Habeshian, Hajnalka E Hartl, Christopher D Hein, Charles W Hutchins, Rachael Jetson, Anthony D Keefe, Hasan Khan, Huan-Qiu Li, Allison Olszewski, Benjamin J Ortiz Cardona, Augustine Osuma, Sanjay C Panchal, Ryan Phelan, Wei Qiu, J Brad Shotwell, Anurupa Shrestha, Myron Srikumaran, Zhi Su, Chaohong Sun, Anup K Upadhyay, Michael D Wood, Haihong Wu, Ruijie K Zhang, Ying Zhang, Gang Zhao, Haizhong Zhu, Matthew P Webster
Discovery of Small Molecule Interleukin 17A Inhibitors with Novel Binding Mode and Stoichiometry: Optimization of DNA-Encoded Chemical Library Hits to In Vivo Active Compounds. Journal of medicinal chemistry 67 (8) (2024)
Ashley L Ramos, Eric R Goedken, Kristine E Frank, Maria A Argiriadi, Sana Bazzaz, Zhiguo Bian, Jesse T C Brown, Paolo A Centrella, Hui-Ju Chen, Jeremy S Disch, Pamela L Donner, David B Duignan, Diana Gikunju, Stephen N Greszler, Marie-Aude Guié, Sevan Habeshian, Hajnalka E Hartl, Christopher D Hein, Charles W Hutchins, Rachael Jetson, Anthony D Keefe, Hasan Khan, Huan-Qiu Li, Allison Olszewski, Benjamin J Ortiz Cardona, Augustine Osuma, Sanjay C Panchal, Ryan Phelan, Wei Qiu, J Brad Shotwell, Anurupa Shrestha, Myron Srikumaran, Zhi Su, Chaohong Sun, Anup K Upadhyay, Michael D Wood, Haihong Wu, Ruijie K Zhang, Ying Zhang, Gang Zhao, Haizhong Zhu, Matthew P Webster
Discovery of Small Molecule Interleukin 17A Inhibitors with Novel Binding Mode and Stoichiometry: Optimization of DNA-Encoded Chemical Library Hits to In Vivo Active Compounds. Journal of medicinal chemistry (2024)
Christopher C Marvin, Stephen N Greszler, Bhadra H Shelat, Eric A Voight
Synthesis of A-9758, an Inverse Agonist of Retinoic Acid-Related Orphan Receptor γt. ACS omega 7 (48) (2022)
Stephen N Greszler, Gang Zhao, Bhadra Shelat, Eric A Voight
Enabling Asymmetric Synthesis of ABBV-3748, a Corrector Compound for the Treatment of Cystic Fibrosis. Organic letters 24 (40) (2022)
Christopher C Marvin, Stephen N Greszler, Bhadra H Shelat, Eric A Voight
Synthesis of A-9758, an Inverse Agonist of Retinoic Acid-Related Orphan Receptor γt. ACS omega 7 (48) (2022)
Marek Buchman, Elliot P Farney, Stephen N Greszler, Robert J Altenbach, Gregory A Gfesser, Eric A Voight
Lithioarene Cycliacylation and Pd-Catalyzed Aminoethylation/Cyclization to Access Electronically Diverse Saturated Isoquinoline Derivatives. The Journal of organic chemistry 87 (1) (2021)
Eric A Voight, Stephen N Greszler, Philip R Kym
Fueling the Pipeline via Innovations in Organic Synthesis. ACS medicinal chemistry letters 12 (9) (2021)
Stephen N Greszler, Gang Zhao, Marek Buchman, Xenia B Searle, Bo Liu, Eric A Voight
General Asymmetric Synthesis of Densely Functionalized Pyrrolidines via Endo-Selective [3+2] Cycloaddition of β-Quaternary-Substituted Nitroalkenes and Azomethine Ylides. The Journal of organic chemistry 85 (11) (2020)
John T Randolph, Eric A Voight, Stephen N Greszler, Brice E Uno, James N Newton, Kenneth M Gleason, DeAnne Stolarik, Cecilia Van Handel, Daniel A J Bow, David A DeGoey
Prodrug Strategies to Improve the Solubility of the HCV NS5A Inhibitor Pibrentasvir (ABT-530). Journal of medicinal chemistry 63 (19) (2020)
Stephen N Greszler, Bhadra Shelat, Eric A Voight
Enabling Synthesis of ABBV-2222, A CFTR Corrector for the Treatment of Cystic Fibrosis. Organic letters 21 (14) (2019)
Eric A Voight, Brian S Brown, Stephen N Greszler, Geoff T Halvorsen, Gang Zhao, Albert W Kruger, John Hartung, Kirill A Lukin, Steven R Martinez, Eric G Moschetta, Michael T Tudesco, Nathan D Ide
Synthesis of ABBV-168, a 2'-Bromouridine for the Treatment of Hepatitis C. The Journal of organic chemistry 84 (8) (2018)
Xueqing Wang, Bo Liu, Xenia Searle, Clinton Yeung, Andrew Bogdan, Stephen N Greszler, Ashvani Singh, Yihong Fan, Andrew M Swensen, Timothy Vortherms, Corina Balut, Ying Jia, Kelly Desino, Wenqing Gao, Hong Yong, Chris Tse, Philip Kym
Discovery of 4-[(2R,4R)-4-({[1-(2,2-Difluoro-1,3-benzodioxol-5-yl)cyclopropyl]carbonyl}amino)-7-(difluoromethoxy)-3,4-dihydro-2H-chromen-2-yl]benzoic Acid (ABBV/GLPG-2222), a Potent Cystic Fibrosis Transmembrane Conductance Regulator (CFTR) Corrector for the Treatment of Cystic Fibrosis. Journal of medicinal chemistry 61 (4) (2018)
Stephen N Greszler, Geoff T Halvorsen, Eric A Voight
Synthesis of Substituted Cyclopropanecarboxylates via Room Temperature Palladium-Catalyzed α-Arylation of Reformatsky Reagents. Organic letters 19 (10) (2017)

Stephen N Greszler.css-eqlu8i{font-size:small;padding-left:4px;} (Stephen Greszler)

Publication Activity (10 Years)

Top Topics

Top Venues

Stephen N Greszler (Stephen Greszler)