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Kinetic characteristics of propofol-induced inhibition of electron-transfer chain and fatty acid oxidation in human and rodent skeletal and cardiac muscles.

Tomáš UrbanPetr WaldaufAdéla KrajčováKateřina JiroutkováMilada HalačováValér DžupaLibor JanoušekEva PokornáFrantišek Duška
Published in: PloS one (2019)
In human skeletal and heart muscle homogenates, propofol in concentrations that are achieved in propofol-anaesthetized patients, causes a direct inhibition of fatty acid oxidation, in addition to inhibiting flux of electrons through inner mitochondrial membrane. The inhibition is more marked in human as compared to rodent tissues.
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