Giacomo Pepe

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 17

Top Topics

Molecular Docking

Botulinum Toxin

Anti Inflammatory

Top Venues

Journal of medicinal chemistry

Oxidative medicine and cellular longevity

This page only lists publications with an associated author ORCID identifier.

Publications

Vincenzo Vestuto, Tania Ciaglia, Simona Musella, Veronica Di Sarno, Gerardina Smaldone, Francesca Di Matteo, Maria Carmina Scala, Valeria Napolitano, Maria Rosaria Miranda, Giuseppina Amodio, Sara Novi, Giacomo Pepe, Manuela Giovanna Basilicata, Erica Gazzillo, Simona Pace, Isabel Maria Gomez-Monterrey, Marina Sala, Giuseppe Bifulco, Mario Felice Tecce, Pietro Campiglia, Carmine Ostacolo, Gianluigi Lauro, Michele Manfra, Alessia Bertamino
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors. Journal of medicinal chemistry (2024)
Nunzio Iraci, Lidia Carotenuto, Tania Ciaglia, Giorgio Belperio, Francesca Di Matteo, Ilaria Mosca, Giusy Carleo, Manuela Giovanna Basilicata, Paolo Ambrosino, Rita Turcio, Deborah Puzo, Giacomo Pepe, Isabel Maria Gomez-Monterrey, Maria Virginia Soldovieri, Veronica Di Sarno, Pietro Campiglia, Francesco Miceli, Alessia Bertamino, Carmine Ostacolo, Taglialatela Maurizio
In Silico Assisted Identification, Synthesis, and In Vitro Pharmacological Characterization of Potent and Selective Blockers of the Epilepsy-Associated KCNT1 Channel. Journal of medicinal chemistry 67 (11) (2024)
Vincenzo Vestuto, Tania Ciaglia, Simona Musella, Veronica Di Sarno, Gerardina Smaldone, Francesca Di Matteo, Maria Carmina Scala, Valeria Napolitano, Maria Rosaria Miranda, Giuseppina Amodio, Sara Novi, Giacomo Pepe, Manuela Giovanna Basilicata, Erica Gazzillo, Simona Pace, Isabel Maria Gomez-Monterrey, Marina Sala, Giuseppe Bifulco, Mario Felice Tecce, Pietro Campiglia, Carmine Ostacolo, Gianluigi Lauro, Michele Manfra, Alessia Bertamino
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors. Journal of medicinal chemistry 67 (15) (2024)
Vincenzo Vestuto, Tania Ciaglia, Simona Musella, Veronica Di Sarno, Gerardina Smaldone, Francesca Di Matteo, Maria Carmina Scala, Valeria Napolitano, Maria Rosaria Miranda, Giuseppina Amodio, Sara Novi, Giacomo Pepe, Manuela Giovanna Basilicata, Erica Gazzillo, Simona Pace, Isabel Maria Gomez-Monterrey, Marina Sala, Giuseppe Bifulco, Mario Felice Tecce, Pietro Campiglia, Carmine Ostacolo, Gianluigi Lauro, Michele Manfra, Alessia Bertamino
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors. Journal of medicinal chemistry 67 (15) (2024)
Nunzio Iraci, Lidia Carotenuto, Tania Ciaglia, Giorgio Belperio, Francesca Di Matteo, Ilaria Mosca, Giusy Carleo, Manuela Giovanna Basilicata, Paolo Ambrosino, Rita Turcio, Deborah Puzo, Giacomo Pepe, Isabel Maria Gomez-Monterrey, Maria Virginia Soldovieri, Veronica Di Sarno, Pietro Campiglia, Francesco Miceli, Alessia Bertamino, Carmine Ostacolo, Taglialatela Maurizio
In Silico Assisted Identification, Synthesis, and In Vitro Pharmacological Characterization of Potent and Selective Blockers of the Epilepsy-Associated KCNT1 Channel. Journal of medicinal chemistry 67 (11) (2024)
Vincenzo Vestuto, Tania Ciaglia, Simona Musella, Veronica Di Sarno, Gerardina Smaldone, Francesca Di Matteo, Maria Carmina Scala, Valeria Napolitano, Maria Rosaria Miranda, Giuseppina Amodio, Sara Novi, Giacomo Pepe, Manuela Giovanna Basilicata, Erica Gazzillo, Simona Pace, Isabel Maria Gomez-Monterrey, Marina Sala, Giuseppe Bifulco, Mario Felice Tecce, Pietro Campiglia, Carmine Ostacolo, Gianluigi Lauro, Michele Manfra, Alessia Bertamino
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors. Journal of medicinal chemistry 67 (15) (2024)
Nunzio Iraci, Lidia Carotenuto, Tania Ciaglia, Giorgio Belperio, Francesca Di Matteo, Ilaria Mosca, Giusy Carleo, Manuela Giovanna Basilicata, Paolo Ambrosino, Rita Turcio, Deborah Puzo, Giacomo Pepe, Isabel Maria Gomez-Monterrey, Maria Virginia Soldovieri, Veronica Di Sarno, Pietro Campiglia, Francesco Miceli, Alessia Bertamino, Carmine Ostacolo, Taglialatela Maurizio
In Silico Assisted Identification, Synthesis, and In Vitro Pharmacological Characterization of Potent and Selective Blockers of the Epilepsy-Associated KCNT1 Channel. Journal of medicinal chemistry 67 (11) (2024)
Nunzio Iraci, Lidia Carotenuto, Tania Ciaglia, Giorgio Belperio, Francesca Di Matteo, Ilaria Mosca, Giusy Carleo, Manuela Giovanna Basilicata, Paolo Ambrosino, Rita Turcio, Deborah Puzo, Giacomo Pepe, Isabel Maria Gomez-Monterrey, Maria Virginia Soldovieri, Veronica Di Sarno, Pietro Campiglia, Francesco Miceli, Alessia Bertamino, Carmine Ostacolo, Taglialatela Maurizio
In Silico Assisted Identification, Synthesis, and In Vitro Pharmacological Characterization of Potent and Selective Blockers of the Epilepsy-Associated KCNT1 Channel. Journal of medicinal chemistry (2024)
Vincenzo Vestuto, Tania Ciaglia, Simona Musella, Veronica Di Sarno, Gerardina Smaldone, Francesca Di Matteo, Maria Carmina Scala, Valeria Napolitano, Maria Rosaria Miranda, Giuseppina Amodio, Sara Novi, Giacomo Pepe, Manuela Giovanna Basilicata, Erica Gazzillo, Simona Pace, Isabel Maria Gomez-Monterrey, Marina Sala, Giuseppe Bifulco, Mario Felice Tecce, Pietro Campiglia, Carmine Ostacolo, Gianluigi Lauro, Michele Manfra, Alessia Bertamino
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors. Journal of medicinal chemistry 67 (15) (2024)
Simona Musella, Danilo D'Avino, Lukas Klaus Peltner, Veronica Di Sarno, Ida Cerqua, Fabrizio Merciai, Vincenzo Vestuto, Tania Ciaglia, Gerardina Smaldone, Francesca Di Matteo, Simone Di Micco, Valeria Napolitano, Giuseppe Bifulco, Giacomo Pepe, Eduardo Maria Sommella, Manuela Giovanna Basilicata, Giovanna Aquino, Isabel Maria Gomez-Monterrey, Pietro Campiglia, Carmine Ostacolo, Fiorentina Roviezzo, Oliver Werz, Antonietta Rossi, Alessia Bertamino
Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis. Journal of medicinal chemistry (2023)
Ida Cerqua, Simona Musella, Lukas Klaus Peltner, Danilo D'Avino, Veronica Di Sarno, Elisabetta Granato, Vincenzo Vestuto, Rita Di Matteo, Simona Pace, Tania Ciaglia, Rossella Bilancia, Gerardina Smaldone, Francesca Di Matteo, Simone Di Micco, Giuseppe Bifulco, Giacomo Pepe, Manuela Giovanna Basilicata, Manuela Rodriquez, Isabel Maria Gomez-Monterrey, Pietro Campiglia, Carmine Ostacolo, Fiorentina Roviezzo, Oliver Werz, Antonietta Rossi, Alessia Bertamino
Discovery and Optimization of Indoline-Based Compounds as Dual 5-LOX/sEH Inhibitors: In Vitro and In Vivo Anti-Inflammatory Characterization. Journal of medicinal chemistry 65 (21) (2022)
Simona Musella, Lidia Carotenuto, Nunzio Iraci, Giulia Baroli, Tania Ciaglia, Piera Nappi, Manuela Giovanna Basilicata, Emanuela Salviati, Vincenzo Barrese, Vincenzo Vestuto, Giuseppe Pignataro, Giacomo Pepe, Eduardo Sommella, Veronica Di Sarno, Michele Manfra, Pietro Campiglia, Isabel Maria Gomez-Monterrey, Alessia Bertamino, Taglialatela Maurizio, Carmine Ostacolo, Francesco Miceli
Beyond Retigabine: Design, Synthesis, and Pharmacological Characterization of a Potent and Chemically Stable Neuronal Kv7 Channel Activator with Anticonvulsant Activity. Journal of medicinal chemistry 65 (16) (2022)
Alessandra Cipriano, Ciro Milite, Alessandra Feoli, Monica Viviano, Giacomo Pepe, Pietro Campiglia, Giuliana Sarno, Sarah Picaud, Satomi Imaide, Nikolai Makukhin, Panagis Filippakopoulos, Alessio Ciulli, Sabrina Castellano, Gianluca Sbardella
Discovery of Benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain. ChemMedChem 17 (20) (2022)
Alessia Bertamino, Carmine Ostacolo, Alicia Medina, Veronica Di Sarno, Gianluigi Lauro, Tania Ciaglia, Vincenzo Vestuto, Giacomo Pepe, Manuela Giovanna Basilicata, Simona Musella, Gerardina Smaldone, Claudia Cristiano, Sara Gonzalez-Rodriguez, Asia Fernandez-Carvajal, Giuseppe Bifulco, Pietro Campiglia, Isabel Maria Gomez-Monterrey, Roberto Russo
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their In Vitro Characterization and In Vivo Analgesic Activities. Journal of medicinal chemistry 63 (17) (2020)
Giacomo Pepe, Manuela Giovanna Basilicata, Albino Carrizzo, Simona Adesso, Carmine Ostacolo, Marina Sala, Eduardo Sommella, Marco Ruocco, Stella Cascioferro, Mariateresa Ambrosio, Simona Pisanti, Veronica Di Sarno, Alessia Bertamino, Stefania Marzocco, Carmine Vecchione, Pietro Campiglia
β-Lactoglobulin Heptapeptide Reduces Oxidative Stress in Intestinal Epithelial Cells and Angiotensin II-Induced Vasoconstriction on Mouse Mesenteric Arteries by Induction of Nuclear Factor Erythroid 2-Related Factor 2 (Nrf2) Translocation. Oxidative medicine and cellular longevity 2019 (2019)
Carmine Ostacolo, Francesco Miceli, Veronica Di Sarno, Piera Nappi, Nunzio Iraci, Maria Virginia Soldovieri, Tania Ciaglia, Paolo Ambrosino, Vincenzo Vestuto, Anna Lauritano, Simona Musella, Giacomo Pepe, Manuela Giovanna Basilicata, Michele Manfra, Diego Romano Perinelli, Ettore Novellino, Alessia Bertamino, Isabel Maria Gomez-Monterrey, Pietro Campiglia, Taglialatela Maurizio
Synthesis and Pharmacological Characterization of Conformationally Restricted Retigabine Analogues as Novel Neuronal Kv7 Channel Activators. Journal of medicinal chemistry 63 (1) (2019)
Marina Sala, Antonia Spensiero, Maria Carmina Scala, Giacomo Pepe, Anna Bilotta, Francesco Paduano, Sabrina D'Agostino, Delia Lanzillotta, Alessia Bertamino, Ettore Novellino, Francesco Trapasso, Isabel M Gomez-Monterrey, Pietro Campiglia
Design, Synthesis, Biological Activity, and Structural Analysis of Lactam-Constrained PTPRJ Agonist Peptides. ChemMedChem 13 (16) (2018)