Gianni Chessari

ORCID

Publication Activity (10 Years)

Years Active: 2021-2024
Publications (10 Years): 13

Top Venues

Journal of medicinal chemistry

RSC medicinal chemistry

Chemical science

ACS central science

This page only lists publications with an associated author ORCID identifier.

Publications

James E H Day, Valerio Berdini, Joan Castro, Gianni Chessari, Thomas G Davies, Philip J Day, Jeffrey D St Denis, Hideto Fujiwara, Satoshi Fukaya, Christopher C F Hamlett, Keisha Hearn, Steven D Hiscock, Rhian S Holvey, Satoru Ito, Navrohit Kandola, Yasuo Kodama, John W Liebeschuetz, Vanessa Martins, Kenichi Matsuo, Paul N Mortenson, Sandra Muench, Yoko Nakatsuru, Hiroaki Ochiiwa, Nicholas Palmer, Torren Peakman, Amanda Price, Michael Reader, David C Rees, Sharna J Rich, Alpesh Shah, Yoshihiro Shibata, Tomoko Smyth, David G Twigg, Nicola G Wallis, Glyn Williams, Nicola E Wilsher, Andrew Woodhead, Tadashi Shimamura, Christopher N Johnson
Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase-2 (SHP2). Journal of medicinal chemistry 67 (6) (2024)
James E H Day, Valerio Berdini, Joan Castro, Gianni Chessari, Thomas G Davies, Philip J Day, Jeffrey D St Denis, Hideto Fujiwara, Satoshi Fukaya, Christopher C F Hamlett, Keisha Hearn, Steven D Hiscock, Rhian S Holvey, Satoru Ito, Navrohit Kandola, Yasuo Kodama, John W Liebeschuetz, Vanessa Martins, Kenichi Matsuo, Paul N Mortenson, Sandra Muench, Yoko Nakatsuru, Hiroaki Ochiiwa, Nicholas Palmer, Torren Peakman, Amanda Price, Michael Reader, David C Rees, Sharna J Rich, Alpesh Shah, Yoshihiro Shibata, Tomoko Smyth, David G Twigg, Nicola G Wallis, Glyn Williams, Nicola E Wilsher, Andrew Woodhead, Tadashi Shimamura, Christopher N Johnson
Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase-2 (SHP2). Journal of medicinal chemistry (2024)
Nick Palmer, Christopher Agnew, Caroline Benn, William J Buffham, Joan N Castro, Gianni Chessari, Mellissa Clark, Benjamin D Cons, Joseph E Coyle, Lee A Dawson, Christopher C F Hamlett, Charlotte Hodson, Finn Holding, Christopher N Johnson, John W Liebeschuetz, Pravin Mahajan, James M McCarthy, Christopher W Murray, Marc O'Reilly, Torren Peakman, Amanda Price, Magdalini Rapti, Judith Reeks, Patrick Schöpf, Jeffrey D St Denis, Chiara Valenzano, Nicola G Wallis, Reto Walser, Heather Weir, Nicola E Wilsher, Andrew Woodhead, Carla F Bento, Dominic Tisi
Fragment-Based Discovery of a Series of Allosteric-Binding Site Modulators of β-Glucocerebrosidase. Journal of medicinal chemistry 67 (13) (2024)
Nick Palmer, Christopher Agnew, Caroline Benn, William J Buffham, Joan N Castro, Gianni Chessari, Mellissa Clark, Benjamin D Cons, Joseph E Coyle, Lee A Dawson, Christopher C F Hamlett, Charlotte Hodson, Finn Holding, Christopher N Johnson, John W Liebeschuetz, Pravin Mahajan, James M McCarthy, Christopher W Murray, Marc O'Reilly, Torren Peakman, Amanda Price, Magdalini Rapti, Judith Reeks, Patrick Schöpf, Jeffrey D St Denis, Chiara Valenzano, Nicola G Wallis, Reto Walser, Heather Weir, Nicola E Wilsher, Andrew Woodhead, Carla F Bento, Dominic Tisi
Fragment-Based Discovery of a Series of Allosteric-Binding Site Modulators of β-Glucocerebrosidase. Journal of medicinal chemistry (2024)
Nick Palmer, Christopher Agnew, Caroline Benn, William J Buffham, Joan N Castro, Gianni Chessari, Mellissa Clark, Benjamin D Cons, Joseph E Coyle, Lee A Dawson, Christopher C F Hamlett, Charlotte Hodson, Finn Holding, Christopher N Johnson, John W Liebeschuetz, Pravin Mahajan, James M McCarthy, Christopher W Murray, Marc O'Reilly, Torren Peakman, Amanda Price, Magdalini Rapti, Judith Reeks, Patrick Schöpf, Jeffrey D St Denis, Chiara Valenzano, Nicola G Wallis, Reto Walser, Heather Weir, Nicola E Wilsher, Andrew Woodhead, Carla F Bento, Dominic Tisi
Fragment-Based Discovery of a Series of Allosteric-Binding Site Modulators of β-Glucocerebrosidase. Journal of medicinal chemistry 67 (13) (2024)
James E H Day, Valerio Berdini, Joan Castro, Gianni Chessari, Thomas G Davies, Philip J Day, Jeffrey D St Denis, Hideto Fujiwara, Satoshi Fukaya, Christopher C F Hamlett, Keisha Hearn, Steven D Hiscock, Rhian S Holvey, Satoru Ito, Navrohit Kandola, Yasuo Kodama, John W Liebeschuetz, Vanessa Martins, Kenichi Matsuo, Paul N Mortenson, Sandra Muench, Yoko Nakatsuru, Hiroaki Ochiiwa, Nicholas Palmer, Torren Peakman, Amanda Price, Michael Reader, David C Rees, Sharna J Rich, Alpesh Shah, Yoshihiro Shibata, Tomoko Smyth, David G Twigg, Nicola G Wallis, Glyn Williams, Nicola E Wilsher, Andrew Woodhead, Tadashi Shimamura, Christopher N Johnson
Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase-2 (SHP2). Journal of medicinal chemistry 67 (6) (2024)
Chloe Townley, Davide Branduardi, Gianni Chessari, Benjamin D Cons, Charlotte Griffiths-Jones, Richard J Hall, Christopher N Johnson, Yuji Ochi, Stuart Whibley, Rachel Grainger
Enabling synthesis in fragment-based drug discovery (FBDD): microscale high-throughput optimisation of the medicinal chemist's toolbox reactions. RSC medicinal chemistry 14 (12) (2023)
Chloe Townley, Davide Branduardi, Gianni Chessari, Benjamin D Cons, Charlotte Griffiths-Jones, Richard J Hall, Christopher N Johnson, Yuji Ochi, Stuart Whibley, Rachel Grainger
Enabling synthesis in fragment-based drug discovery (FBDD): microscale high-throughput optimisation of the medicinal chemist's toolbox reactions. RSC medicinal chemistry 14 (12) (2023)
Connor J Taylor, Kobi C Felton, Daniel S Wigh, Mohammed I Jeraal, Rachel Grainger, Gianni Chessari, Christopher N Johnson, Alexei A Lapkin
Accelerated Chemical Reaction Optimization Using Multi-Task Learning. ACS central science 9 (5) (2023)
Jeffrey D St Denis, Gianni Chessari, Anne Cleasby, Benjamin D Cons, Suzanna Cowan, Samuel E Dalton, Charlotte East, Christopher W Murray, Marc O'Reilly, Torren Peakman, Magdalini Rapti, Jessie L Stow
X-ray Screening of an Electrophilic Fragment Library and Application toward the Development of a Novel ERK 1/2 Covalent Inhibitor. Journal of medicinal chemistry 65 (18) (2022)
Benjamin D Cons, David G Twigg, Rajendra Kumar, Gianni Chessari
Electrostatic Complementarity in Structure-Based Drug Design. Journal of medicinal chemistry 65 (11) (2022)
Gianni Chessari, Rachel Grainger, Rhian S Holvey, R Frederick Ludlow, Paul N Mortenson, David C Rees
C-H functionalisation tolerant to polar groups could transform fragment-based drug discovery (FBDD). Chemical science 12 (36) (2021)
Gianni Chessari, Ian R Hardcastle, Jong Sook Ahn, Burcu Anil, Elizabeth Anscombe, Ruth H Bawn, Luke D Bevan, Timothy J Blackburn, Ildiko Buck, Celine Cano, Benoit Carbain, Juan Castro, Ben Cons, Sarah J Cully, Jane A Endicott, Lynsey Fazal, Bernard T Golding, Roger J Griffin, Karen Haggerty, Suzannah J Harnor, Keisha Hearn, Stephen Hobson, Rhian S Holvey, Steven Howard, Claire E Jennings, Christopher N Johnson, John Lunec, Duncan C Miller, David R Newell, Martin E M Noble, Judith Reeks, Charlotte H Revill, Christiane Riedinger, Jeffrey D St Denis, Emiliano Tamanini, Huw Thomas, Neil T Thompson, Mladen Vinković, Stephen R Wedge, Pamela A Williams, Nicola E Wilsher, Bian Zhang, Yan Zhao
Structure-Based Design of Potent and Orally Active Isoindolinone Inhibitors of MDM2-p53 Protein-Protein Interaction. Journal of medicinal chemistry 64 (7) (2021)

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Publication Activity (10 Years)

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Gianni Chessari