Michael P Pollastri

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 23

Top Venues

Journal of medicinal chemistry

ACS infectious diseases

PLoS neglected tropical diseases

RSC medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Lori Ferrins, Rosario Diaz, Carlos Cordon-Obras, Domingo Rojas-Barros, Antonio Quotadamo, Daniel P Oehme, Gloria Ceballos-Pérez, Uma Swaminathan, Guiomar Pérez-Moreno, Cristina Bosch-Navarrete, Raquel García-Hernández, Claudia Gomez-Liñan, Andreu Saura, Luis Miguel Ruiz-Perez, Francisco Gamarro, Maria Santos Martinez-Martinez, Pilar Manzano, Dolores Gonzalez Pacanowska, Miguel Navarro, Michael P Pollastri
Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei . Journal of medicinal chemistry 67 (16) (2024)
Lori Ferrins, Rosario Diaz, Carlos Cordon-Obras, Domingo Rojas-Barros, Antonio Quotadamo, Daniel P Oehme, Gloria Ceballos-Pérez, Uma Swaminathan, Guiomar Pérez-Moreno, Cristina Bosch-Navarrete, Raquel García-Hernández, Claudia Gomez-Liñan, Andreu Saura, Luis Miguel Ruiz-Perez, Francisco Gamarro, Maria Santos Martinez-Martinez, Pilar Manzano, Dolores Gonzalez Pacanowska, Miguel Navarro, Michael P Pollastri
Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei . Journal of medicinal chemistry 67 (16) (2024)
Lori Ferrins, Rosario Diaz, Carlos Cordon-Obras, Domingo Rojas-Barros, Antonio Quotadamo, Daniel P Oehme, Gloria Ceballos-Pérez, Uma Swaminathan, Guiomar Pérez-Moreno, Cristina Bosch-Navarrete, Raquel García-Hernández, Claudia Gomez-Liñan, Andreu Saura, Luis Miguel Ruiz-Perez, Francisco Gamarro, Maria Santos Martinez-Martinez, Pilar Manzano, Dolores Gonzalez Pacanowska, Miguel Navarro, Michael P Pollastri
Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei . Journal of medicinal chemistry (2024)
Lori Ferrins, Rosario Diaz, Carlos Cordon-Obras, Domingo Rojas-Barros, Antonio Quotadamo, Daniel P Oehme, Gloria Ceballos-Pérez, Uma Swaminathan, Guiomar Pérez-Moreno, Cristina Bosch-Navarrete, Raquel García-Hernández, Claudia Gomez-Liñan, Andreu Saura, Luis Miguel Ruiz-Perez, Francisco Gamarro, Maria Santos Martinez-Martinez, Pilar Manzano, Dolores Gonzalez Pacanowska, Miguel Navarro, Michael P Pollastri
Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei . Journal of medicinal chemistry 67 (16) (2024)
Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K Gadekar, Brady Greene, Michael Chichioco, Carlos E Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P Pollastri
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of medicinal chemistry (2023)
Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K Gadekar, Brady Greene, Michael Chichioco, Carlos E Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P Pollastri
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of medicinal chemistry 66 (3) (2023)
Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K Gadekar, Brady Greene, Michael Chichioco, Carlos E Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P Pollastri
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of medicinal chemistry 66 (3) (2023)
Maria Dichiara, Quillon J Simpson, Antonio Quotadamo, Hitesh B Jalani, Anson X Huang, Caroline C Millard, Dana M Klug, Edwin G Tse, Matthew H Todd, Daniel Gedder Silva, Flavio da Silva Emery, J Eric Carlson, Shao Liang Zheng, Margot Vleminckx, An Matheeussen, Guy Caljon, Michael P Pollastri, Peter Sjö, Benjamin G Perry, Lori Ferrins
Structure-Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis. ACS infectious diseases (2023)
Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K Gadekar, Brady Greene, Michael Chichioco, Carlos E Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P Pollastri
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of medicinal chemistry 66 (3) (2023)
Jing Chai, Christopher C Arico-Muendel, Yun Ding, Michael P Pollastri, Sarah Scott, Mark A Mantell, Gang Yao
Synthesis of a DNA-Encoded Macrocyclic Library Utilizing Intramolecular Benzimidazole Formation. Bioconjugate chemistry (2023)
Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K Gadekar, Brady Greene, Michael Chichioco, Carlos E Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P Pollastri
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of medicinal chemistry 66 (3) (2023)
Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K Gadekar, Brady Greene, Michael Chichioco, Carlos E Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P Pollastri
Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of medicinal chemistry 66 (3) (2023)
Dana M Klug, Eftychia M Mavrogiannaki, Katherine C Forbes, Lisseth Silva, Rosario Diaz-Gonzalez, Guiomar Pérez-Moreno, Gloria Ceballos-Pérez, Raquel Garcia-Hernández, Cristina Bosch-Navarrete, Carlos Cordón-Obras, Claudia Gómez-Liñán, Andreu Saura, Jeremiah D Momper, Maria Santos Martinez-Martinez, Pilar Manzano, Ali Syed, Nelly El-Sakkary, Conor R Caffrey, Francisco Gamarro, Luis Miguel Ruiz-Perez, Dolores Gonzalez Pacanowska, Lori Ferrins, Miguel Navarro, Michael P Pollastri
Lead Optimization of 3,5-Disubstituted-7-Azaindoles for the Treatment of Human African Trypanosomiasis. Journal of medicinal chemistry 64 (13) (2021)
Dana M Klug, Rosario Diaz-Gonzalez, Travis J DeLano, Eftychia M Mavrogiannaki, Melissa J Buskes, Raeann M Dalton, John K Fisher, Katherine M Schneider, Vivian Hilborne, Melanie G Fritsche, Quillon J Simpson, Westley F Tear, William G Devine, Guiomar Pérez-Moreno, Gloria Ceballos-Pérez, Raquel García-Hernández, Cristina Bosch-Navarrete, Luis Miguel Ruiz-Pérez, Francisco Gamarro, Dolores González-Pacanowska, Maria Santos Martinez-Martinez, Pilar Manzano-Chinchon, Miguel Navarro, Michael P Pollastri, Lori Ferrins
Structure-property studies of an imidazoquinoline chemotype with antitrypanosomal activity. RSC medicinal chemistry 11 (8) (2020)
Westley F Tear, Seema Bag, Rosario Diaz-Gonzalez, Gloria Ceballos-Pérez, Domingo I Rojas-Barros, Carlos Cordon-Obras, Guiomar Pérez-Moreno, Raquel García-Hernández, Maria Santos Martinez-Martinez, Luis Miguel Ruiz-Perez, Francisco Gamarro, Dolores Gonzalez Pacanowska, Conor R Caffrey, Lori Ferrins, Pilar Manzano, Miguel Navarro, Michael P Pollastri
Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5-b]pyridazines for the Treatment of Human African Trypanosomiasis. Journal of medicinal chemistry 63 (2) (2020)
Baljinder Singh, Rosario Diaz-Gonzalez, Gloria Ceballos-Perez, Domingo I Rojas-Barros, Naresh Gunaganti, Kirsten Gillingwater, Maria Santos Martinez-Martinez, Pilar Manzano, Miguel Navarro, Michael P Pollastri
Medicinal Chemistry Optimization of a Diaminopurine Chemotype: Toward a Lead for Trypanosoma brucei Inhibitors. Journal of medicinal chemistry 63 (17) (2020)
Kelly A Bachovchin, Amrita Sharma, Seema Bag, Dana M Klug, Katherine M Schneider, Baljinder Singh, Hitesh B Jalani, Melissa J Buskes, Naimee Mehta, Scott Tanghe, Jeremiah D Momper, Richard J Sciotti, Ana Rodriguez, Kojo Mensa-Wilmot, Michael P Pollastri, Lori Ferrins
Improvement of Aqueous Solubility of Lapatinib-Derived Analogues: Identification of a Quinolinimine Lead for Human African Trypanosomiasis Drug Development. Journal of medicinal chemistry 62 (2) (2019)
Dana M Klug, Rosario Diaz-Gonzalez, Guiomar Pérez-Moreno, Gloria Ceballos-Pérez, Raquel García-Hernández, Veronica Gomez-Pérez, Luis Miguel Ruiz-Pérez, Domingo I Rojas-Barros, Francisco Gamarro, Dolores González-Pacanowska, María S Martínez-Martínez, Pilar Manzano, Lori Ferrins, Conor R Caffrey, Miguel Navarro, Michael P Pollastri
Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents. PLoS neglected tropical diseases 13 (2) (2019)
Dana M Klug, Laura Tschiegg, Rosario Diaz, Domingo Rojas-Barros, Guiomar Perez-Moreno, Gloria Ceballos, Raquel García-Hernández, Maria Santos Martinez-Martinez, Pilar Manzano, Luis Miguel Ruiz, Conor R Caffrey, Francisco Gamarro, Dolores Gonzalez Pacanowska, Lori Ferrins, Miguel Navarro, Michael P Pollastri
Hit-to-Lead Optimization of Benzoxazepinoindazoles As Human African Trypanosomiasis Therapeutics. Journal of medicinal chemistry 63 (5) (2019)
Lori Ferrins, Amrita Sharma, Sarah M Thomas, Naimee Mehta, Jessey Erath, Scott Tanghe, Susan E Leed, Ana Rodriguez, Kojo Mensa-Wilmot, Richard J Sciotti, Kirsten Gillingwater, Michael P Pollastri
Anilinoquinoline based inhibitors of trypanosomatid proliferation. PLoS neglected tropical diseases 12 (11) (2018)
Naimee Mehta, Lori Ferrins, Susan E Leed, Richard J Sciotti, Michael P Pollastri
Optimization of Physicochemical Properties for 4-Anilinoquinoline Inhibitors of Plasmodium falciparum Proliferation. ACS infectious diseases 4 (4) (2018)
William G Devine, Rosario Diaz-Gonzalez, Gloria Ceballos-Perez, Domingo Rojas, Takashi Satoh, Westley Tear, Ranae M Ranade, Ximena Barros-Álvarez, Wim G J Hol, Frederick S Buckner, Miguel Navarro, Michael P Pollastri
From Cells to Mice to Target: Characterization of NEU-1053 (SB-443342) and Its Analogues for Treatment of Human African Trypanosomiasis. ACS infectious diseases 3 (3) (2017)
Lori Ferrins, Michael P Pollastri
The Importance of Collaboration between Industry, Academics, and Nonprofits in Tropical Disease Drug Discovery. ACS infectious diseases 4 (4) (2017)

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Publication Activity (10 Years)

Top Topics

Top Venues

Michael P Pollastri