Thomas Stockner

ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 51

Top Venues

Nature communications

Proceedings of the National Academy of Sciences of the United States of America

eLife

Journal of neurochemistry

Medical University of Vienna

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Medical University of Vienna Dec 01 2018

Austria

Assoc. Prof. :: Pharmacology

Medical University of Vienna Dec 01 2015 - Nov 30 2018

Austria

Assistant Professor :: Institute of Pharmacology

Medical University of Vienna May 01 2014 - Nov 30 2015

Austria

Univ. Ass. :: Pharamcology

Medical University of Vienna Jan 01 2010 - Apr 30 2014

Austria

Post Doc :: Pharmacology

Austrian Institute of Technology Apr 01 2008 - Jun 30 2010

Austria

Group leader :: Bioresources

Austrian Institute of Technology Oct 10 2005 - Mar 01 2008

Austria

Application Scientist :: Bioresources

University of Calgary Jan 01 2003 - Oct 01 2005

Canada

Post Doc :: Biological Sciences

University of Graz Jul 01 2001 - Dec 31 2002

Austria

Post Doc :: Chemistry

Publications

Ralph Gradisch, Katharina Schlögl, Erika Lazzarin, Marco Niello, Julian Maier, Felix P Mayer, Leticia Alves da Silva, Sophie M C Skopec, Randy D Blakely, Harald H Sitte, Marko D Mihovilovic, Thomas Stockner
Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors. Nature communications 15 (1) (2024)
Leticia Alves da Silva, Erika Lazzarin, Ralph Gradisch, Amy Clarke, Thomas Stockner
Free energy profile of the substrate-induced occlusion of the human serotonin transporter. Journal of neurochemistry (2024)
Ana Sofia Alberto-Silva, Selina Hemmer, Hailey A Bock, Leticia Alves da Silva, Kenneth R Scott, Nina Kastner, Manan Bhatt, Marco Niello, Kathrin Jäntsch, Oliver Kudlacek, Elena Bossi, Thomas Stockner, Markus R Meyer, John D McCorvy, Simon D Brandt, Pierce V Kavanagh, Harald H Sitte
Bioisosteric analogs of MDMA: Improving the pharmacological profile? Journal of neurochemistry (2024)
Amy Clarke, Julia Skerjanz, Matthias A F Gsell, Patrick Wiedner, Hazel Erkan-Candag, Klaus Groschner, Thomas Stockner, Oleksandra Tiapko
PIP 2 modulates TRPC3 activity via TRP helix and S4-S5 linker. Nature communications 15 (1) (2024)
Ralph Gradisch, Katharina Schlögl, Erika Lazzarin, Marco Niello, Julian Maier, Felix P Mayer, Leticia Alves da Silva, Sophie M C Skopec, Randy D Blakely, Harald H Sitte, Marko D Mihovilovic, Thomas Stockner
Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors. Nature communications 15 (1) (2024)
Ana Sofia Alberto-Silva, Selina Hemmer, Hailey A Bock, Leticia Alves da Silva, Kenneth R Scott, Nina Kastner, Manan Bhatt, Marco Niello, Kathrin Jäntsch, Oliver Kudlacek, Elena Bossi, Thomas Stockner, Markus R Meyer, John D McCorvy, Simon D Brandt, Pierce V Kavanagh, Harald H Sitte
Bioisosteric analogs of MDMA with improved pharmacological profile. bioRxiv : the preprint server for biology (2024)
Ralph Gradisch, Katharina Schlögl, Erika Lazzarin, Marco Niello, Julian Maier, Felix P Mayer, Leticia Alves da Silva, Sophie M C Skopec, Randy D Blakely, Harald H Sitte, Marko D Mihovilovic, Thomas Stockner
Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors. Nature communications 15 (1) (2024)
Ana Sofia Alberto-Silva, Selina Hemmer, Hailey A Bock, Leticia Alves da Silva, Kenneth R Scott, Nina Kastner, Manan Bhatt, Marco Niello, Kathrin Jäntsch, Oliver Kudlacek, Elena Bossi, Thomas Stockner, Markus R Meyer, John D McCorvy, Simon D Brandt, Pierce V Kavanagh, Harald H Sitte
Bioisosteric analogs of MDMA: Improving the pharmacological profile? Journal of neurochemistry (2024)
Ralph Gradisch, Katharina Schlögl, Erika Lazzarin, Marco Niello, Julian Maier, Felix P Mayer, Leticia Alves da Silva, Sophie M C Skopec, Randy D Blakely, Harald H Sitte, Marko D Mihovilovic, Thomas Stockner
Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors. Nature communications 15 (1) (2024)
Ana Sofia Alberto-Silva, Selina Hemmer, Hailey A Bock, Leticia Alves da Silva, Kenneth R Scott, Nina Kastner, Manan Bhatt, Marco Niello, Kathrin Jäntsch, Oliver Kudlacek, Elena Bossi, Thomas Stockner, Markus R Meyer, John D McCorvy, Simon D Brandt, Pierce V Kavanagh, Harald H Sitte
Bioisosteric analogs of MDMA with improved pharmacological profile. bioRxiv : the preprint server for biology (2024)
Ana Sofia Alberto-Silva, Selina Hemmer, Hailey A Bock, Leticia Alves da Silva, Kenneth R Scott, Nina Kastner, Manan Bhatt, Marco Niello, Kathrin Jäntsch, Oliver Kudlacek, Elena Bossi, Thomas Stockner, Markus R Meyer, John D McCorvy, Simon D Brandt, Pierce V Kavanagh, Harald H Sitte
Bioisosteric analogs of MDMA with improved pharmacological profile. bioRxiv : the preprint server for biology (2024)
Amy Clarke, Julia Skerjanz, Matthias A F Gsell, Patrick Wiedner, Hazel Erkan-Candag, Klaus Groschner, Thomas Stockner, Oleksandra Tiapko
PIP 2 modulates TRPC3 activity via TRP helix and S4-S5 linker. Nature communications 15 (1) (2024)
Amy Clarke, Julia Skerjanz, Matthias A F Gsell, Patrick Wiedner, Hazel Erkan-Candag, Klaus Groschner, Thomas Stockner, Oleksandra Tiapko
PIP 2 modulates TRPC3 activity via TRP helix and S4-S5 linker. Nature communications 15 (1) (2024)
Ralph Gradisch, Katharina Schlögl, Erika Lazzarin, Marco Niello, Julian Maier, Felix P Mayer, Leticia Alves da Silva, Sophie M C Skopec, Randy D Blakely, Harald H Sitte, Marko D Mihovilovic, Thomas Stockner
Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors. Nature communications 15 (1) (2024)
Ana Sofia Alberto-Silva, Selina Hemmer, Hailey A Bock, Leticia Alves da Silva, Kenneth R Scott, Nina Kastner, Manan Bhatt, Marco Niello, Kathrin Jäntsch, Oliver Kudlacek, Elena Bossi, Thomas Stockner, Markus R Meyer, John D McCorvy, Simon D Brandt, Pierce V Kavanagh, Harald H Sitte
Bioisosteric analogs of MDMA: Improving the pharmacological profile? Journal of neurochemistry (2024)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Zsuzsanna Gyöngy, Gábor Mocsár, Éva Hegedűs, Thomas Stockner, Zsuzsanna Ritter, László Homolya, Anita Schamberger, Tamás I Orbán, Judit Remenyik, Gergely Szakacs, Katalin Goda
Nucleotide binding is the critical regulator of ABCG2 conformational transitions. eLife 12 (2023)
Kornel Ozvoldik, Thomas Stockner, Elmar Krieger
YASARA Model-Interactive Molecular Modeling from Two Dimensions to Virtual Realities. Journal of chemical information and modeling (2023)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Amy Clarke, Clemens V Farr, Ali El-Kasaby, Daniel Szöllősi, Michael Freissmuth, Sonja Sucic, Thomas Stockner
Probing binding and occlusion of substrate in the human creatine transporter-1 by computation and mutagenesis. Protein science : a publication of the Protein Society (2023)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Zsuzsanna Gyöngy, Gábor Mocsár, Éva Hegedűs, Thomas Stockner, Zsuzsanna Ritter, László Homolya, Anita Schamberger, Tamás I Orbán, Judit Remenyik, Gergely Szakacs, Katalin Goda
Nucleotide binding is the critical regulator of ABCG2 conformational transitions. eLife 12 (2023)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Zsuzsanna Gyöngy, Gábor Mocsár, Éva Hegedűs, Thomas Stockner, Zsuzsanna Ritter, László Homolya, Anita Schamberger, Tamás I Orbán, Judit Remenyik, Gergely Szakacs, Katalin Goda
Nucleotide binding is the critical regulator of ABCG2 conformational transitions. eLife 12 (2023)
Zsuzsanna Gyöngy, Gábor Mocsár, Éva Hegedűs, Thomas Stockner, Zsuzsanna Ritter, László Homolya, Anita Schamberger, Tamás I Orbán, Judit Remenyik, Gergely Szakacs, Katalin Goda
Nucleotide binding is the critical regulator of ABCG2 conformational transitions. eLife 12 (2023)
Zsuzsanna Gyöngy, Gábor Mocsár, Éva Hegedűs, Thomas Stockner, Zsuzsanna Ritter, László Homolya, Anita Schamberger, Tamás I Orbán, Judit Remenyik, Gergely Szakacs, Katalin Goda
Nucleotide binding is the critical regulator of ABCG2 conformational transitions. eLife 12 (2023)
Marco Niello, Spyridon Sideromenos, Ralph Gradisch, Ronan O Shea, Jakob Schwazer, Julian Maier, Nina Kastner, Walter Sandtner, Kathrin Jäntsch, Carl R Lupica, Alexander F Hoffman, Gert Lubec, Claus J Løland, Thomas Stockner, Daniela D Pollak, Michael H Baumann, Harald H Sitte
Persistent binding at dopamine transporters determines sustained psychostimulant effects. Proceedings of the National Academy of Sciences of the United States of America 120 (6) (2023)
Zsuzsanna Gyöngy, Gábor Mocsár, Éva Hegedűs, Thomas Stockner, Zsuzsanna Ritter, László Homolya, Anita Schamberger, Tamás I Orbán, Judit Remenyik, Gergely Szakacs, Katalin Goda
Nucleotide binding is the critical regulator of ABCG2 conformational transitions. eLife 12 (2023)
Hazel Erkan-Candag, Denis Krivic, Matthias A F Gsell, Mina Aleksanyan, Thomas Stockner, Rumiana Dimova, Oleksandra Tiapko, Klaus Groschner
Characterization of DAG Binding to TRPC Channels by Target-Dependent cis-trans Isomerization of OptoDArG. Biomolecules 12 (6) (2022)
Dániel Szöllősi, Thomas Stockner
Sodium Binding Stabilizes the Outward-Open State of SERT by Limiting Bundle Domain Motions. Cells 11 (2) (2022)
Hazel Erkan-Candag, Amy Clarke, Oleksandra Tiapko, Matthias A F Gsell, Thomas Stockner, Klaus Groschner
Diacylglycerols interact with the L2 lipidation site in TRPC3 to induce a sensitized channel state. EMBO reports 23 (7) (2022)
Basavraj Khanppnavar, Julian Maier, Freja Herborg, Ralph Gradisch, Erika Lazzarin, Dino Luethi, Jae-Won Yang, Chao Qi, Marion Holy, Kathrin Jäntsch, Oliver Kudlacek, Klaus Schicker, Thomas M Werge, Ulrik Gether, Thomas Stockner, Volodymyr M Korkhov, Harald H Sitte
Structural basis of organic cation transporter-3 inhibition. Nature communications 13 (1) (2022)
Amy Clarke, Klaus Groschner, Thomas Stockner
Exploring TRPC3 Interaction with Cholesterol through Coarse-Grained Molecular Dynamics Simulations. Biomolecules 12 (7) (2022)
Muhammad Imran Sohail, Yaprak Donmez Cakil, Dániel Szöllősi, Thomas Stockner, Peter Chiba
The Bile Salt Export Pump: Molecular Structure, Study Models and Small-Molecule Drugs for the Treatment of Inherited BSEP Deficiencies. International journal of molecular sciences 22 (2) (2021)
Kornel Ozvoldik, Thomas Stockner, Burkhard Rammner, Elmar Krieger
Assembly of Biomolecular Gigastructures and Visualization with the Vulkan Graphics API. Journal of chemical information and modeling 61 (10) (2021)
Markus Ponleitner, Daniel Szöllösi, Ali El-Kasaby, Florian Koban, Michael Freissmuth, Thomas Stockner
Thermal unfolding of the human serotonin transporter: differential effect by stabilizing and destabilizing mutations and cholesterol on thermodynamic and kinetic stability. Molecular pharmacology (2021)
James I Mitchell-White, Thomas Stockner, Nicholas D Holliday, Stephen J Briddon, Ian D Kerr
Analysis of Sequence Divergence in Mammalian ABCGs Predicts a Structural Network of Residues That Underlies Functional Divergence. International journal of molecular sciences 22 (6) (2021)
Deborah Rudin, John D McCorvy, Grant C Glatfelter, Dino Luethi, Dániel Szöllősi, Tea Ljubišić, Pierce V Kavanagh, Geraldine Dowling, Marion Holy, Kathrin Jaentsch, Donna Walther, Simon D Brandt, Thomas Stockner, Michael H Baumann, Adam L Halberstadt, Harald H Sitte
(2-Aminopropyl)benzo[β]thiophenes (APBTs) are novel monoamine transporter ligands that lack stimulant effects but display psychedelic-like activity in mice. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology (2021)
Thomas Stockner, Ralph Gradisch, Lutz Schmitt
The role of the degenerate nucleotide binding site in type I ABC exporters. FEBS letters 594 (23) (2020)
Dániel Szöllősi, Peter Chiba, Gergely Szakacs, Thomas Stockner
Conversion of chemical to mechanical energy by the nucleotide binding domains of ABCB1. Scientific reports 10 (1) (2020)
Kumaresan Jayaraman, Anand K Das, Dino Luethi, Dániel Szöllősi, Gerhard J Schütz, Maarten E A Reith, Harald H Sitte, Thomas Stockner
SLC6 transporter oligomerization. Journal of neurochemistry 157 (4) (2020)
Shahrooz Nasrollahi-Shirazi, Daniel Szöllösi, Qiong Yang, Edin Muratspahic, Ali El-Kasaby, Sonja Sucic, Thomas Stockner, Christian Nanoff, Michael Freissmuth
Functional Impact of the G279S Substitution in the Adenosine A1-Receptor (A1R-G279S7.44), a Mutation Associated with Parkinson's Disease. Molecular pharmacology 98 (3) (2020)
Narakorn Khunweeraphong, James I Mitchell-White, Dániel Szöllősi, Toka O K Hussein, Karl Kuchler, Ian D Kerr, Thomas Stockner, Jyh-Yeuan Lee
Picky ABCG5/G8 and promiscuous ABCG2 - a tale of fatty diets and drug toxicity. FEBS letters 594 (23) (2020)
Anand Kant Das, Oliver Kudlacek, Florian Baumgart, Kathrin Jaentsch, Thomas Stockner, Harald H Sitte, Gerhard J Schütz
Dopamine transporter forms stable dimers in the live cell plasma membrane in a phosphatidylinositol 4,5-bisphosphate-independent manner. The Journal of biological chemistry 294 (14) (2019)
Narakorn Khunweeraphong, Daniel Szöllősi, Thomas Stockner, Karl Kuchler
The ABCG2 multidrug transporter is a pump gated by a valve and an extracellular lid. Nature communications 10 (1) (2019)
Jawad A Khan, Azmat Sohail, Kumaresan Jayaraman, Dániel Szöllősi, Walter Sandtner, Harald H Sitte, Thomas Stockner
The Amino Terminus of LeuT Changes Conformation in an Environment Sensitive Manner. Neurochemical research 45 (6) (2019)
Nicholas G Campbell, Aparna Shekar, Jenny I Aguilar, Dungeng Peng, Vikas Navratna, Dongxue Yang, Alexander N Morley, Amanda M Duran, Greta Galli, Brian O'Grady, Ramnarayan Ramachandran, James S Sutcliffe, Harald H Sitte, Kevin Erreger, Jens Meiler, Thomas Stockner, Leon M Bellan, Heinrich J G Matthies, Eric Gouaux, Hassane S Mchaourab, Aurelio Galli
Structural, functional, and behavioral insights of dopamine dysfunction revealed by a deletion in SLC6A3. Proceedings of the National Academy of Sciences of the United States of America 116 (9) (2019)
Nechama Silverstein, Alaa Sliman, Thomas Stockner, Baruch I Kanner
Both reentrant loops of the sodium-coupled glutamate transporters contain molecular determinants of cation selectivity. The Journal of biological chemistry 293 (37) (2018)
Kumaresan Jayaraman, Alex N Morley, Dániel Szöllősi, Tsjerk A Wassenaar, Harald H Sitte, Thomas Stockner
Dopamine transporter oligomerization involves the scaffold domain, but spares the bundle domain. PLoS computational biology 14 (6) (2018)

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Publication Activity (10 Years)

Top Topics

Top Venues

Thomas Stockner