Open-Label, Multicenter, Phase I/II, First-in-Human Trial of TK216: A First-Generation EWS::FLI1 Fusion Protein Antagonist in Ewing Sarcoma.
Paul A MeyersNoah FedermanNajat C DawPeter M AndersonLara E DavisAeRang KimMargaret E MacyAngela PietrofesoRavin RatanRichard F RiedelMatteo TruccoJames B BreitmeyerJeffrey A ToretskyJoseph A LudwigPublished in: Journal of clinical oncology : official journal of the American Society of Clinical Oncology (2024)
TK216 administered as 14-day continuous infusion with or without vincristine was well tolerated and showed limited activity at the RP2D in R/R ES.