Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents
Keyphrases
Publications
volume 33, number 4, 2024
- Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-KangDesign, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
- Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-KangDesign, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
- Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-KangDesign, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
- Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-KangDesign, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
volume 33, number 8, 2024
2023
- Simon D P Baugh, Anna Chaly, Damian G Weaver, David B Whitman, Jeffrey C Pelletier, Haiyan Bian, Katie B Freeman, Allen B Reitz, Richard W ScottAmide- and bis-amide-linked highly potent and broadly active antifungal agents for the treatment of invasive fungal infections- towards the discovery of pre-clinical development candidate FC12406. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents (2023)
- Carolyn D Dzierba, Bireshwar Dasgupta, George Karageorge, Walter Kostich, Brian Hamman, Jason Allen, Kim M Esposito, Ramesh Padmanabha, James Grace, Kimberley Lentz, John Morrison, Daniel Morgan, Amy Easton, Clotilde Bourin, Marc R Browning, Ramkumar Rajamani, Andrew Good, Dawn D Parker, Jodi K Muckelbauer, Javed Khan, Daniel Camac, Kaushik Ghosh, Vivek Halan, Jonathan S Lippy, Kenneth S Santone, R Rex Denton, Ryan Westphal, Linda J Bristow, Charles M Conway, Joanne J Bronson, John E Macor
- Shijia Zhao, Xiaoyan Zhang, Min Tang, Xiaocheng Liu, Jialun Deng, Wei Zhou, Zhi Xu
- Maryam Bayanati, Mona Khoramjouy, Mehrdad Faizi, Mahsa Azami Movahed, Mohammad Mahboubi-Rabbani, Afshin ZarghiNovel Benzo[4,5]imidazo[1,2- a ]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents (2023)
- Priyanka Kashyap, Sangeeta Verma, Pankaj Gupta, Rakesh Narang, Sukhbir Lal, Manish Devgun
- Maryam Bayanati, Mona Khoramjouy, Mehrdad Faizi, Mahsa Azami Movahed, Mohammad Mahboubi-Rabbani, Afshin ZarghiNovel Benzo[4,5]imidazo[1,2- a ]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents (2023)
- Carolyn D Dzierba, Bireshwar Dasgupta, George Karageorge, Walter Kostich, Brian Hamman, Jason Allen, Kim M Esposito, Ramesh Padmanabha, James Grace, Kimberley Lentz, John Morrison, Daniel Morgan, Amy Easton, Clotilde Bourin, Marc R Browning, Ramkumar Rajamani, Andrew Good, Dawn D Parker, Jodi K Muckelbauer, Javed Khan, Daniel Camac, Kaushik Ghosh, Vivek Halan, Jonathan S Lippy, Kenneth S Santone, R Rex Denton, Ryan Westphal, Linda J Bristow, Charles M Conway, Joanne J Bronson, John E Macor
- Shijia Zhao, Xiaoyan Zhang, Min Tang, Xiaocheng Liu, Jialun Deng, Wei Zhou, Zhi Xu
- Maryam Bayanati, Mona Khoramjouy, Mehrdad Faizi, Mahsa Azami Movahed, Mohammad Mahboubi-Rabbani, Afshin ZarghiNovel Benzo[4,5]imidazo[1,2- a ]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents (2023)
- Simon D P Baugh, Anna Chaly, Damian G Weaver, David B Whitman, Jeffrey C Pelletier, Haiyan Bian, Katie B Freeman, Allen B Reitz, Richard W ScottAmide- and bis-amide-linked highly potent and broadly active antifungal agents for the treatment of invasive fungal infections- towards the discovery of pre-clinical development candidate FC12406. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents (2023)
- Maryam Bayanati, Mona Khoramjouy, Mehrdad Faizi, Mahsa Azami Movahed, Mohammad Mahboubi-Rabbani, Afshin ZarghiNovel Benzo[4,5]imidazo[1,2- a ]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents (2023)
- Priyanka Kashyap, Sangeeta Verma, Pankaj Gupta, Rakesh Narang, Sukhbir Lal, Manish Devgun
volume 32, number 3, 2023
- Maryam Bayanati, Mona Khoramjouy, Mehrdad Faizi, Mahsa Azami Movahed, Mohammad Mahboubi-Rabbani, Afshin ZarghiNovel Benzo[4,5]imidazo[1,2- a ]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (3) (2023)
- Maryam Bayanati, Mona Khoramjouy, Mehrdad Faizi, Mahsa Azami Movahed, Mohammad Mahboubi-Rabbani, Afshin ZarghiNovel Benzo[4,5]imidazo[1,2- a ]pyrimidine derivatives as selective Cyclooxygenase-2 Inhibitors: Design, synthesis, docking studies, and biological evaluation. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (3) (2023)
volume 32, number 4, 2023
- Shijia Zhao, Xiaoyan Zhang, Min Tang, Xiaocheng Liu, Jialun Deng, Wei Zhou, Zhi Xu
volume 32, number 5, 2023
- Zhen Ye, Tong-Shi-Yao Zhao, Shan-Bin Li, Xian-Li Zhou, Qin Luo, Jiang-Ke Qin, Cheng-Qin Liang, Ping Wang, Guang-Bo Ge
- Mahsa Azami Movahed, Fatemeh Khadem Abbasi, Mahsa Rajabi, Niusha Abedi, Nima Naderi, Bahram Daraei, Afshin ZarghiDesign, synthesis, and biological evaluation of new 2-(4-(methylsulfonyl)phenyl)- N -phenylimidazo[1,2- a ]pyridin-3-amine as selective COX-2 inhibitors. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (5) (2023)
volume 32, number 6, 2023
- Aamer Saeed, Saba Ashraf, Mubashir Aziz, Pervaiz Ali Channar, Syeda Abida Ejaz, Ammara Fayyaz, Qamar Abbas, Fatmah Ali Alasmary, Abdulnasser Mahmoud Karami, Arfa Tehzeeb, Amara Mumtaz, Hesham R El-SeediDesign, synthesis, biochemical and in silico characterization of novel naphthalene-thiourea conjugates as potential and selective inhibitors of alkaline phosphatase. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (6) (2023)
- Duong Ngoc Toan, Nguyen Dinh Thanh, Mai Xuan Truong, Dinh Thuy Van, Nguyen Ngoc ThanhDesign, synthesis, molecular docking study and molecular dynamics simulation of new coumarin-pyrimidine hybrid compounds having anticancer and antidiabetic activity. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (6) (2023)
- Shikha Kaushik, Sarvesh Kumar Paliwal, Malliga R Iyer, Vaishali M Patil
volume 32, number 7, 2023
- Jeffrey Yang, Haifa Albanyan, Yiling Wang, Yanhui Yang, Amrik Sahota, Longqin HuDevelopment of convenient crystallization inhibition assays for structure-activity relationship studies in the discovery of crystallization inhibitors. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (7) (2023)
volume 32, number 2, 2022
- Amgad M Rabie, Mohnad AbdallaEvaluation of a series of nucleoside analogs as effective anticoronaviral-2 drugs against the Omicron-B.1.1.529/BA.2 subvariant: A repurposing research study. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (2) (2022)
- Hezhen Wang, Xun Sun, Chunyong Wei, Jing Wang, Yingshu Xu, Guohui Bai, Qizheng Yao, Lei Zhang
- Amgad M Rabie, Mohnad AbdallaEvaluation of a series of nucleoside analogs as effective anticoronaviral-2 drugs against the Omicron-B.1.1.529/BA.2 subvariant: A repurposing research study. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 32 (2) (2022)
- Hezhen Wang, Xun Sun, Chunyong Wei, Jing Wang, Yingshu Xu, Guohui Bai, Qizheng Yao, Lei Zhang
volume 31, number 3, 2022
- Connor A Lejcher, Eric M Villa, James T Fletcher
volume 31, number 4, 2022
- Qiuchan Wu, Jiang Zeng, Jinfu Dong
- Guoxin Du, Weiwei Du, Yuanlong An, Minnan Wang, Feifei Hao, Xiaochu Tong, Qi Gong, Xiangdong He, Hualiang Jiang, Wei He, Mingyue Zheng, Donglei Zhang
volume 31, number 7, 2022
- Giri R Gnawali, Koichi Okumura, Karolina Perez, Rosa Gallagher, Julia Wulfkuhle, Emanuel F Petricoin, Sathish Kumar Reddy Padi, Jeremiah Bearss, Zhiyong He, Wei Wang, Andrew S Kraft
- Jin-Jin Sun, Jin-Ping Wang, Tian-Ze Li, Yun-Bao Ma, Dong Xue, Ji-Jun Chen
- Haozhou Tan, Chunlong Ma, Jun WangInvalidation of dieckol and 1,2,3,4,6-pentagalloylglucose (PGG) as SARS-CoV-2 main protease inhibitors and the discovery of PGG as a papain-like protease inhibitor. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 31 (7) (2022)
volume 31, number 8, 2022
- Gaofenngwe Nkomba, Gisella Terre'Blanche, Helena D Janse van Rensburg, Lesetja J LegoabeDesign, synthesis and evaluation of amino-3,5-dicyanopyridines and thieno[2,3-b]pyridines as ligands of adenosine A 1 receptors for the potential treatment of epilepsy. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 31 (8) (2022)