Joseph M Salvino (Joseph Salvino)

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 48

Top Topics

Respiratory Syndrome Coronavirus

Angiotensin Converting Enzyme

Transcranial Magnetic Stimulation

Top Venues

ACS chemical biology

Nature communications

Journal of medicinal chemistry

Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents

This page only lists publications with an associated author ORCID identifier.

Publications

Felicite Majoumo-Mbe, Neba Abongwa Sangbong, Alain Tadjong Tcho, Cyril T Namba-Nzanguim, Conrad V Simoben, Donatus Bekindaka Eni, Mustafa A Isa, Adi Narayana Reddy Poli, Joel A Cassel, Joseph M Salvino, Luis J Montaner, Ian Tietjen, Fidele Ntie-Kang
5-chloro-3-(2-(2,4-dinitrophenyl) hydrazono)indolin-2-one: synthesis, characterization, biochemical and computational screening against SARS-CoV-2. Chemicke zvesti 78 (6) (2024)
Marie L Matos-Hernández, Robert M Samples, Grayce Dyer, Victoria M Casimir Montán, Chris A Morales-Colón, Joseph M Salvino, Luis J Montaner, Joel A Cassel, Troy E Messick, Ian Tietjen, Eduardo J E Caro-Diaz
Metabolomic Analysis and Antiviral Screening of a Marine Algae Library Yield Jobosic Acid (2,5-Dimethyltetradecanoic Acid) as a Selective Inhibitor of SARS-CoV-2. Journal of natural products 87 (6) (2024)
Mariana J Shayo, Baraka Samwel, Daniel M Shadrack, Joel A Cassel, Joseph M Salvino, Luis J Montaner, Geradius Deogratias, Ian Tietjen, Lucy Kiruri, Samson Hilonga, Ester Innocent
Drug repositioning identifies salvinorin A and deacetylgedunin (DCG) enriched plant extracts as novel inhibitors of Mpro, RBD-ACE2 and TMPRRS2 proteins. RSC advances 14 (29) (2024)
Adi N R Poli, Ian Tietjen, Nitesh K Nandwana, Joel Cassel, Troy E Messick, Emery T Register, Frederick Keeney, Rajesh Rajaiah, Atul K Verma, Kabita Pandey, Arpan Acharya, Siddappa N Byrareddy, Luis J Montaner, Joseph M Salvino
Design of novel and highly selective SARS-CoV-2 main protease inhibitors. Antimicrobial agents and chemotherapy (2024)
Andreia Cristina Karklin Fontana, Adi N R Poli, Jitendra Gour, Yellamelli V V Srikanth, Nicholas Anastasi, Devipriya Ashok, Apeksha Khatiwada, Katelyn L Reeb, Mary Hongying Cheng, Ivet Bahar, Scott M Rawls, Joseph M Salvino
Synthesis and Structure-Activity Relationships for Glutamate Transporter Allosteric Modulators. Journal of medicinal chemistry (2024)
Mariana J Shayo, Baraka Samwel, Daniel M Shadrack, Joel A Cassel, Joseph M Salvino, Luis J Montaner, Geradius Deogratias, Ian Tietjen, Lucy Kiruri, Samson Hilonga, Ester Innocent
Drug repositioning identifies salvinorin A and deacetylgedunin (DCG) enriched plant extracts as novel inhibitors of Mpro, RBD-ACE2 and TMPRRS2 proteins. RSC advances 14 (29) (2024)
Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-Kang
Design, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology 19 (2) (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology 19 (2) (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology 19 (2) (2024)
Andreia Cristina Karklin Fontana, Adi N R Poli, Jitendra Gour, Yellamelli V V Srikanth, Nicholas Anastasi, Devipriya Ashok, Apeksha Khatiwada, Katelyn L Reeb, Mary Hongying Cheng, Ivet Bahar, Scott M Rawls, Joseph M Salvino
Synthesis and Structure-Activity Relationships for Glutamate Transporter Allosteric Modulators. Journal of medicinal chemistry 67 (8) (2024)
Andreia Cristina Karklin Fontana, Adi N R Poli, Jitendra Gour, Yellamelli V V Srikanth, Nicholas Anastasi, Devipriya Ashok, Apeksha Khatiwada, Katelyn L Reeb, Mary Hongying Cheng, Ivet Bahar, Scott M Rawls, Joseph M Salvino
Synthesis and Structure-Activity Relationships for Glutamate Transporter Allosteric Modulators. Journal of medicinal chemistry (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology 19 (2) (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology 19 (2) (2024)
Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-Kang
Design, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
Marie L Matos-Hernández, Robert M Samples, Grayce Dyer, Victoria M Casimir Montán, Chris A Morales-Colón, Joseph M Salvino, Luis J Montaner, Joel A Cassel, Troy E Messick, Ian Tietjen, Eduardo J E Caro-Diaz
Metabolomic Analysis and Antiviral Screening of a Marine Algae Library Yield Jobosic Acid (2,5-Dimethyltetradecanoic Acid) as a Selective Inhibitor of SARS-CoV-2. Journal of natural products (2024)
Nitesh K Nandwana, Om P S Patel, Manish K Mehra, Anil Kumar, Joseph M Salvino
Recent Advances in Metal-Catalyzed Approaches for the Synthesis of Quinazoline Derivatives. Molecules (Basel, Switzerland) 29 (10) (2024)
Andreia Cristina Karklin Fontana, Adi N R Poli, Jitendra Gour, Yellamelli V V Srikanth, Nicholas Anastasi, Devipriya Ashok, Apeksha Khatiwada, Katelyn L Reeb, Mary Hongying Cheng, Ivet Bahar, Scott M Rawls, Joseph M Salvino
Synthesis and Structure-Activity Relationships for Glutamate Transporter Allosteric Modulators. Journal of medicinal chemistry 67 (8) (2024)
Andreia Cristina Karklin Fontana, Adi N R Poli, Jitendra Gour, Yellamelli V V Srikanth, Nicholas Anastasi, Devipriya Ashok, Apeksha Khatiwada, Katelyn L Reeb, Mary Hongying Cheng, Ivet Bahar, Scott M Rawls, Joseph M Salvino
Synthesis and Structure-Activity Relationships for Glutamate Transporter Allosteric Modulators. Journal of medicinal chemistry 67 (8) (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology (2024)
Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-Kang
Design, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
Marie L Matos-Hernández, Robert M Samples, Grayce Dyer, Victoria M Casimir Montán, Chris A Morales-Colón, Joseph M Salvino, Luis J Montaner, Joel A Cassel, Troy E Messick, Ian Tietjen, Eduardo J E Caro-Diaz
Metabolomic Analysis and Antiviral Screening of a Marine Algae Library Yield Jobosic Acid (2,5-Dimethyltetradecanoic Acid) as a Selective Inhibitor of SARS-CoV-2. Journal of natural products 87 (6) (2024)
Sehbanul Islam, Jitendra Gour, Thomas Beer, Hsin-Yao Tang, Joel Cassel, Joseph M Salvino, Luca Busino
A Tandem-Affinity Purification Method for Identification of Primary Intracellular Drug-Binding Proteins. ACS chemical biology 19 (2) (2024)
Nitesh K Nandwana, Om P S Patel, Manish K Mehra, Anil Kumar, Joseph M Salvino
Recent Advances in Metal-Catalyzed Approaches for the Synthesis of Quinazoline Derivatives. Molecules (Basel, Switzerland) 29 (10) (2024)
Donatus Bekindaka Eni, Joel A Cassel, Cyril T Namba-Nzanguim, Conrad V Simoben, Ian Tietjen, Ravikumar Akunuri, Joseph M Salvino, Fidele Ntie-Kang
Design, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents 33 (4) (2024)
Ali Vaziri-Gohar, Jonathan J Hue, Ata Abbas, Hallie J Graor, Omid Hajihassani, Mehrdad Zarei, George Titomihelakis, John Feczko, Moeez Rathore, Sylwia Chelstowska, Alexander W Loftus, Rui Wang, Mahsa Zarei, Maryam Goudarzi, Renliang Zhang, Belinda Willard, Li Zhang, Adam Kresak, Joseph E Willis, Gi-Ming Wang, Curtis Tatsuoka, Joseph M Salvino, Ilya Bederman, Henri Brunengraber, Costas A Lyssiotis, Jonathan R Brody, Jordan M Winter
Increased glucose availability sensitizes pancreatic cancer to chemotherapy. Nature communications 14 (1) (2023)
Ali Vaziri-Gohar, Jonathan J Hue, Ata Abbas, Hallie J Graor, Omid Hajihassani, Mehrdad Zarei, George Titomihelakis, John Feczko, Moeez Rathore, Sylwia Chelstowska, Alexander W Loftus, Rui Wang, Mahsa Zarei, Maryam Goudarzi, Renliang Zhang, Belinda Willard, Li Zhang, Adam Kresak, Joseph E Willis, Gi-Ming Wang, Curtis Tatsuoka, Joseph M Salvino, Ilya Bederman, Henri Brunengraber, Costas A Lyssiotis, Jonathan R Brody, Jordan M Winter
Increased glucose availability sensitizes pancreatic cancer to chemotherapy. Nature communications 14 (1) (2023)
Ali Vaziri-Gohar, Jonathan J Hue, Ata Abbas, Hallie J Graor, Omid Hajihassani, Mehrdad Zarei, George Titomihelakis, John Feczko, Moeez Rathore, Sylwia Chelstowska, Alexander W Loftus, Rui Wang, Mahsa Zarei, Maryam Goudarzi, Renliang Zhang, Belinda Willard, Li Zhang, Adam Kresak, Joseph E Willis, Gi-Ming Wang, Curtis Tatsuoka, Joseph M Salvino, Ilya Bederman, Henri Brunengraber, Costas A Lyssiotis, Jonathan R Brody, Jordan M Winter
Increased glucose availability sensitizes pancreatic cancer to chemotherapy. Nature communications 14 (1) (2023)
Michael Ippolito, Francesco De Pascali, Nathan Hopfinger, Konstantin E Komolov, Daniela Laurinavichyute, Poli Adi Narayana Reddy, Leon A Sakkal, Kyle Z Rajkowski, Ajay P Nayak, Justin Lee, Jordan Lee, Gaoyuan Cao, Preston S Donover, Melvin Reichman, Steven S An, Joseph M Salvino, Raymond B Penn, Roger S Armen, Charles P Scott, Jeffrey L Benovic
Identification of a β-arrestin-biased negative allosteric modulator for the β 2 -adrenergic receptor. Proceedings of the National Academy of Sciences of the United States of America 120 (31) (2023)
Ali Vaziri-Gohar, Jonathan J Hue, Ata Abbas, Hallie J Graor, Omid Hajihassani, Mehrdad Zarei, George Titomihelakis, John Feczko, Moeez Rathore, Sylwia Chelstowska, Alexander W Loftus, Rui Wang, Mahsa Zarei, Maryam Goudarzi, Renliang Zhang, Belinda Willard, Li Zhang, Adam Kresak, Joseph E Willis, Gi-Ming Wang, Curtis Tatsuoka, Joseph M Salvino, Ilya Bederman, Henri Brunengraber, Costas A Lyssiotis, Jonathan R Brody, Jordan M Winter
Increased glucose availability sensitizes pancreatic cancer to chemotherapy. Nature communications 14 (1) (2023)
Yange Cui, Luyang Wang, Qingbao Ding, Jihae Shin, Joel Cassel, Jingjing Liu, Joseph M Salvino, Bin Tian
Elevated pre-mRNA 3' end processing activity in cancer cells renders vulnerability to inhibition of cleavage and polyadenylation. Nature communications 14 (1) (2023)
Ali Vaziri-Gohar, Jonathan J Hue, Ata Abbas, Hallie J Graor, Omid Hajihassani, Mehrdad Zarei, George Titomihelakis, John Feczko, Moeez Rathore, Sylwia Chelstowska, Alexander W Loftus, Rui Wang, Mahsa Zarei, Maryam Goudarzi, Renliang Zhang, Belinda Willard, Li Zhang, Adam Kresak, Joseph E Willis, Gi-Ming Wang, Curtis Tatsuoka, Joseph M Salvino, Ilya Bederman, Henri Brunengraber, Costas A Lyssiotis, Jonathan R Brody, Jordan M Winter
Increased glucose availability sensitizes pancreatic cancer to chemotherapy. Nature communications 14 (1) (2023)
Clare M Adams, Ramkrishna Mitra, You-Cai Xiao, Peter Michener, Juan Palazzo, Allen Chao, Jitendra Gour, Joel A Cassel, Joseph M Salvino, Christine M Eischen
Targeted MDM2 degradation reveals a new vulnerability for p53 inactivated triple negative breast cancer. Cancer discovery (2023)
Clare M Adams, Ramkrishna Mitra, You-Cai Xiao, Peter Michener, Juan Palazzo, Allen Chao, Jitendra Gour, Joel A Cassel, Joseph M Salvino, Christine M Eischen
Targeted MDM2 degradation reveals a new vulnerability for p53 inactivated triple negative breast cancer. Cancer discovery (2023)
Katelyn D Miller, Seamus O'Connor, Katherine A Pniewski, Toshitha Kannan, Reyes Acosta, Gauri Mirji, Sara Papp, Michael Hulse, Dzmitry Mukha, Sabina I Hlavaty, Kelsey N Salcido, Fabrizio Bertolazzi, Yellamelli V V Srikanth, Steven Zhao, Kathryn E Wellen, Rahul S Shinde, Daniel T Claiborne, Andrew Kossenkov, Joseph M Salvino, Zachary T Schug
Acetate acts as a metabolic immunomodulator by bolstering T-cell effector function and potentiating antitumor immunity in breast cancer. Nature cancer (2023)
Luke Invernizzi, Phanankosi Moyo, Joel A Cassel, Freddie J Isaacs, Joseph M Salvino, Luis J Montaner, Ian Tietjen, Vinesh J Maharaj
Use of hyphenated analytical techniques to identify the bioactive constituents of Gunnera perpensa L., a South African medicinal plant, which potently inhibit SARS-CoV-2 spike glycoprotein-host ACE2 binding. Analytical and bioanalytical chemistry 414 (13) (2022)
Ali Vaziri-Gohar, Joel Cassel, Farheen S Mohammed, Mehrdad Zarei, Jonathan J Hue, Omid Hajihassani, Hallie J Graor, Yellamelli V V Srikanth, Saadia A Karim, Ata Abbas, Erin Prendergast, Vanessa Chen, Erryk S Katayama, Katerina Dukleska, Imran Khokhar, Anthony Andren, Li Zhang, Chunying Wu, Bernadette Erokwu, Chris A Flask, Mahsa Zarei, Rui Wang, Luke D Rothermel, Andrea M P Romani, Jessica Bowers, Robert Getts, Curtis Tatsuoka, Jennifer P Morton, Ilya Bederman, Henri Brunengraber, Costas Andreas Lyssiotis, Joseph M Salvino, Jonathan R Brody, Jordan M Winter
Limited nutrient availability in the tumor microenvironment renders pancreatic tumors sensitive to allosteric IDH1 inhibitors. Nature cancer 3 (7) (2022)
Jagadish C Ghosh, Michela Perego, Ekta Agarwal, Irene Bertolini, Yuan Wang, Aaron R Goldman, Hsin-Yao Tang, Andrew V Kossenkov, Catherine J Landis, Lucia R Languino, Edward F Plow, Annamaria Morotti, Luisa Ottobrini, Marco Locatelli, David W Speicher, M Cecilia Caino, Joel Cassel, Joseph M Salvino, Marie E Robert, Valentina Vaira, Dario C Altieri
Ghost mitochondria drive metastasis through adaptive GCN2/Akt therapeutic vulnerability. Proceedings of the National Academy of Sciences of the United States of America 119 (8) (2022)
Shaili Aggarwal, Mary Hongying Cheng, Joseph M Salvino, Ivet Bahar, Ole Valente Mortensen
Functional Characterization of the Dopaminergic Psychostimulant Sydnocarb as an Allosteric Modulator of the Human Dopamine Transporter. Biomedicines 9 (6) (2021)
Hongzhuang Peng, Joel Cassel, Daniel S McCracken, Jeremy W Prokop, Eleonora Sementino, Mitchell Cheung, Paul R Collop, Alexander Polo, Surbhi Joshi, Jacob P Mandell, Kasirajan Ayyanathan, David Hinds, S Bruce Malkowicz, J William Harbour, Anne M Bowcock, Joseph M Salvino, Eileen J Kennedy, Joseph R Testa, Frank J Rauscher
Kinetic Characterization of ASXL1/2-Mediated Allosteric Regulation of the BAP1 Deubiquitinase. Molecular cancer research : MCR 19 (7) (2021)
Jianglan Liu, Vito W Rebecca, Andrew V Kossenkov, Thomas Connelly, Jingjing Liu, Alexis Gutierrez, Min Xiao, Ling Li, Gao Zhang, Anastasia Samarkina, Delaine Zayasbazan, Jie Zhang, Chaoran Cheng, Zhi Wei, Gretchen M Alicea, Mizuho Fukunaga-Kalabis, Clemens Krepler, Pedro Aza-Blanc, Chih-Cheng Yang, Bela Delvadia, Cynthia Tong, Ye Huang, Maya Delvadia, Alice S Morias, Katrin Sproesser, Patricia Brafford, Joshua X Wang, Marilda Beqiri, Rajasekharan Somasundaram, Adina Vultur, Denitsa M Hristova, Lawrence W Wu, Yiling Lu, Gordon B Mills, Wei Xu, Giorgos C Karakousis, George X Xu, Lynn M Schuchter, Tara C Mitchell, Ravi K Amaravadi, Lawrence N Kwong, Dennie T Frederick, Genevieve Marie Boland, Joseph M Salvino, David W Speicher, Keith T Flaherty, Ze'ev A Ronai, Meenhard Herlyn
Neural Crest-Like Stem Cell Transcriptome Analysis Identifies LPAR1 in Melanoma Progression and Therapy Resistance. Cancer research 81 (20) (2021)
Katelyn D Miller, Katherine Pniewski, Caroline E Perry, Sara B Papp, Joshua D Shaffer, Jesse N Velasco-Silva, Jessica C Casciano, Tomas M Aramburu, Yellamelli V V Srikanth, Joel Cassel, Emmanuel Skordalakes, Andrew V Kossenkov, Joseph M Salvino, Zachary T Schug
Targeting ACSS2 with a Transition-State Mimetic Inhibits Triple-Negative Breast Cancer Growth. Cancer research 81 (5) (2021)
Zachary E Stine, Zachary T Schug, Joseph M Salvino, Chi Van Dang
Targeting cancer metabolism in the era of precision oncology. Nature reviews. Drug discovery (2021)
Patrizia Porazzi, Marco De Dominici, Joseph M Salvino, Bruno Calabretta
Targeting the CDK6 Dependence of Ph+ Acute Lymphoblastic Leukemia. Genes 12 (9) (2021)
Christopher W Schultz, Grace A McCarthy, Teena Nerwal, Avinoam Nevler, James B DuHadaway, Matthew D McCoy, Wei Jiang, Samantha Z Brown, Austin Goetz, Aditi Jain, Valerie S Calvert, Vikalp Vishwakarma, Dezhen Wang, Ranjan Preet, Joel Cassel, Ross Summer, Hoora Shaghaghi, Yves Pommier, Simone A Baechler, Michael J Pishvaian, Talia Golan, Charles J Yeo, Emanuel F Petricoin, George C Prendergast, Joseph M Salvino, Pankaj K Singh, Dan A Dixon, Jonathan R Brody
The FDA-Approved Anthelmintic Pyrvinium Pamoate Inhibits Pancreatic Cancer Cells in Nutrient-Depleted Conditions by Targeting the Mitochondria. Molecular cancer therapeutics 20 (11) (2021)
Thibaut Barnoud, Jessica C Leung, Julia I-Ju Leu, Subhasree Basu, Adi Narayana Reddy Poli, Joshua L D Parris, Alexandra Indeglia, Tetyana Martynyuk, Madeline Good, Keerthana Gnanapradeepan, Emilio Sanseviero, Rebecca Moeller, Hsin-Yao Tang, Joel Cassel, Andrew V Kossenkov, Jingjing Liu, David W Speicher, Dmitry I Gabrilovich, Joseph M Salvino, Donna L George, Maureen E Murphy
A Novel Inhibitor of HSP70 Induces Mitochondrial Toxicity and Immune Cell Recruitment in Tumors. Cancer research 80 (23) (2020)
Kumar Sachin Singh, Rishabh Sharma, Poli Adi Narayana Reddy, Prashanthi Vonteddu, Madeline Good, Anjana Sundarrajan, Hyeree Choi, Kar Muthumani, Andrew Kossenkov, Aaron R Goldman, Hsin-Yao Tang, Maxim Totrov, Joel Cassel, Maureen E Murphy, Rajasekharan Somasundaram, Meenhard Herylyn, Joseph M Salvino, Farokh Dotiwala
IspH inhibitors kill Gram-negative bacteria and mobilize immune clearance. Nature 589 (7843) (2020)
Nadezhda Tikhmyanova, Steve Tutton, Kayla A Martin, Fang Lu, Andrew V Kossenkov, Nicholas Paparoidamis, Shannon Kenney, Joseph M Salvino, Paul M Lieberman
Small molecule perturbation of the CAND1-Cullin1-ubiquitin cycle stabilizes p53 and triggers Epstein-Barr virus reactivation. PLoS pathogens 13 (7) (2017)