Ian Collins

Publication Activity (10 Years)

Years Active: 2016-2023
Publications (10 Years): 15

Top Topics

Fluorescence Imaging

Protein Protein

Endoplasmic Reticulum Stress

Top Venues

Journal of medicinal chemistry

Cancer research

Journal of proteome research

Scientific reports

This page only lists publications with an associated author ORCID identifier.

Publications

François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry 66 (4) (2023)
François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry 66 (4) (2023)
François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry 66 (4) (2023)
François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry (2023)
François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry 66 (4) (2023)
François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry 66 (4) (2023)
François Saint-Dizier, Thomas P Matthews, Aaron M Gregson, Hugues Prevet, Tatiana McHardy, Giampiero Colombano, Harry Saville, Martin Rowlands, Caroline Ewens, Peter Craig McAndrew, Kathy Tomlin, Delphine Guillotin, Grace Wing-Yan Mak, Konstantinos Drosopoulos, Ioannis Poursaitidis, Rosemary Burke, Rob van Montfort, Spiros Linardopoulos, Ian Collins
Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes. Journal of medicinal chemistry 66 (4) (2023)
Fernando J Sialana, Theodoros I Roumeliotis, Habib Bouguenina, Laura Chan Wah Hak, Hannah Wang, John Caldwell, Ian Collins, Rajesh Chopra, Jyoti S Choudhary
SimPLIT: Simplified Sample Preparation for Large-Scale Isobaric Tagging Proteomics. Journal of proteome research 21 (8) (2022)
Suzanne O'Connor, Yann-Vaï Le Bihan, Isaac M Westwood, Manjuan Liu, Oi Wei Mak, Gabriel Zazeri, Ana Paula Ribeiro Povinelli, Alan M Jones, Rob van Montfort, Jóhannes Reynisson, Ian Collins
Discovery and Characterization of a Cryptic Secondary Binding Site in the Molecular Chaperone HSP70. Molecules (Basel, Switzerland) 27 (3) (2022)
Nicola Lockwood, Silvia Martini, Ainara Lopez-Pardo, Katharina Deiss, Hendrika A Segeren, Robert K Semple, Ian Collins, Dimitra Repana, Mathias Cobbaut, Tanya N Soliman, Francesca Ciccarelli, Peter J Parker
Genome-Protective Topoisomerase 2a-Dependent G2 Arrest Requires p53 in hTERT-Positive Cancer Cells. Cancer research 82 (9) (2022)
Rebecca F Rogers, Michael I Walton, Daniel L Cherry, Ian Collins, Paul Andrew Clarke, Michelle D Garrett, Paul Workman
CHK1 Inhibition Is Synthetically Lethal with Loss of B-Family DNA Polymerase Function in Human Lung and Colorectal Cancer Cells. Cancer research 80 (8) (2020)
Giampiero Colombano, John J Caldwell, Thomas P Matthews, Chitra Bhatia, Amar Joshi, Tatiana McHardy, Ngai Yi Mok, Yvette Newbatt, Lisa Pickard, Jade Strover, Somaieh Hedayat, Michael I Walton, Stephanie M Myers, Alan M Jones, Harry Saville, Craig McAndrew, Rosemary Burke, Suzanne A Eccles, Faith E Davies, Richard Bayliss, Ian Collins
Binding to an Unusual Inactive Kinase Conformation by Highly Selective Inhibitors of Inositol-Requiring Enzyme 1α Kinase-Endoribonuclease. Journal of medicinal chemistry 62 (5) (2019)
Katie Pollock, Manjuan Liu, Mariola Zaleska, Mirco Meniconi, Mark Pfuhl, Ian Collins, Sebastian Guettler
Fragment-based screening identifies molecules targeting the substrate-binding ankyrin repeat domains of tankyrase. Scientific reports 9 (1) (2019)
Nicola E A Chessum, Swee Y Sharp, John J Caldwell, A Elisa Pasqua, Birgit Wilding, Giampiero Colombano, Ian Collins, Bugra Ozer, Meirion Richards, Martin Rowlands, Mark Stubbs, Rosemary Burke, P Craig McAndrew, Paul Andrew Clarke, Paul Workman, Matthew D Cheeseman, Keith Jones
Demonstrating In-Cell Target Engagement Using a Pirin Protein Degradation Probe (CCT367766). Journal of medicinal chemistry 61 (3) (2018)
Stuart S Rankin, John J Caldwell, Nora B Cronin, Rob L M van Montfort, Ian Collins
Synthesis of a Ribose-Incorporating Medium Ring Scaffold via a Challenging Ring-Closing Metathesis Reaction. European journal of organic chemistry 2016 (26) (2016)