Maikel Wijtmans

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 17

Top Topics

Silver Nanoparticles

Wastewater Treatment

Fluorescent Probe

Top Venues

Molecules (Basel, Switzerland)

Journal of medicinal chemistry

Angewandte Chemie (International ed. in English)

Pharmaceuticals (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Yang Zheng, Meichun Gao, Maikel Wijtmans, Henry F Vischer, Rob Leurs
Synthesis and Pharmacological Characterization of New Photocaged Agonists for Histamine H 3 and H 4 Receptors. Pharmaceuticals (Basel, Switzerland) 17 (4) (2024)
Yang Zheng, Meichun Gao, Maikel Wijtmans, Henry F Vischer, Rob Leurs
Synthesis and Pharmacological Characterization of New Photocaged Agonists for Histamine H 3 and H 4 Receptors. Pharmaceuticals (Basel, Switzerland) 17 (4) (2024)
Tom Dekker, Jaap W Harteveld, Gábor Wágner, Max C M de Vries, Hans Custers, Andrea C van de Stolpe, Iwan J P de Esch, Maikel Wijtmans
Green Drug Discovery: Novel Fragment Space from the Biomass-Derived Molecule Dihydrolevoglucosenone (Cyrene TM ). Molecules (Basel, Switzerland) 28 (4) (2023)
Tom Dekker, Mathilde A C H Janssen, Christina Sutherland, Rene W M Aben, Hans W Scheeren, Daniel Blanco-Ania, Floris P J T Rutjes, Maikel Wijtmans, Iwan J P de Esch
An Automated, Open-Source Workflow for the Generation of (3D) Fragment Libraries. ACS medicinal chemistry letters 14 (5) (2023)
Icaro A Simon, Evert J Homan, Maikel Wijtmans, Michael Sundström, Rob Leurs, Iwan J P de Esch, Barbara A Zarzycka
PSW-Designer: An Open-Source Computational Platform for the Design and Virtual Screening of Photopharmacological Ligands. Journal of chemical information and modeling (2023)
Tom Dekker, Jaap W Harteveld, Gábor Wágner, Max C M de Vries, Hans Custers, Andrea C van de Stolpe, Iwan J P de Esch, Maikel Wijtmans
Green Drug Discovery: Novel Fragment Space from the Biomass-Derived Molecule Dihydrolevoglucosenone (Cyrene TM ). Molecules (Basel, Switzerland) 28 (4) (2023)
Tom Dekker, Mathilde A C H Janssen, Christina Sutherland, Rene W M Aben, Hans W Scheeren, Daniel Blanco-Ania, Floris P J T Rutjes, Maikel Wijtmans, Iwan J P de Esch
An Automated, Open-Source Workflow for the Generation of (3D) Fragment Libraries. ACS medicinal chemistry letters 14 (5) (2023)
Tom Dekker, Jaap W Harteveld, Gábor Wágner, Max C M de Vries, Hans Custers, Andrea C van de Stolpe, Iwan J P de Esch, Maikel Wijtmans
Green Drug Discovery: Novel Fragment Space from the Biomass-Derived Molecule Dihydrolevoglucosenone (Cyrene TM ). Molecules (Basel, Switzerland) 28 (4) (2023)
Tom Dekker, Jaap W Harteveld, Gábor Wágner, Max C M de Vries, Hans Custers, Andrea C van de Stolpe, Iwan J P de Esch, Maikel Wijtmans
Green Drug Discovery: Novel Fragment Space from the Biomass-Derived Molecule Dihydrolevoglucosenone (Cyrene TM ). Molecules (Basel, Switzerland) 28 (4) (2023)
David J Hamilton, Marieke Beemsterboer, Caroline M Carter, Jasmina Elsayed, Rilana E M Huiberts, Hanna F Klein, Peter O'Brien, Iwan J P de Esch, Maikel Wijtmans
Puckering the Planar Landscape of Fragments: Design and Synthesis of a 3D Cyclobutane Fragment Library. ChemMedChem 17 (9) (2022)
Zhiyong Wang, Reggie Bosma, Sebastiaan Kuhne, Jelle van den Bor, Wrej Garabitian, Henry F Vischer, Maikel Wijtmans, Rob Leurs, Iwan J P de Esch
Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics. ACS omega 6 (19) (2021)
Xavier Gómez-Santacana, Sabrina M de Munnik, Tamara A M Mocking, Niels J Hauwert, Shanliang Sun, Prashanna Vijayachandran, Iwan J P de Esch, Henry F Vischer, Maikel Wijtmans, Rob Leurs
A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light. Beilstein journal of organic chemistry 15 (2019)
Niels J Hauwert, Tamara A M Mocking, Daniel P DA Costa, Ken Lion, Yara Huppelschoten, Henry F Vischer, Iwan J P De Esch, Maikel Wijtmans, Rob Leurs
A Photoswitchable Agonist for the Histamine H3 Receptor, a Prototypic Family A G-Protein-Coupled Receptor. Angewandte Chemie (International ed. in English) 58 (14) (2019)
Reggie Bosma, Zhiyong Wang, Albert Jelke Kooistra, Nick Bushby, Sebastiaan Kuhne, Jelle van den Bor, Michael J Waring, Chris de Graaf, Iwan J de Esch, Henry F Vischer, Robert J Sheppard, Maikel Wijtmans, Rob Leurs
Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine. Journal of medicinal chemistry 62 (14) (2019)
Gábor Wágner, Tamara A M Mocking, Marta Arimont, Gustavo Provensi, Barbara Rani, Bruna Silva-Marques, Gniewomir Latacz, Daniel Da Costa Pereira, Christina Karatzidou, Henry F Vischer, Maikel Wijtmans, Katarzyna Kieć-Kononowicz, Iwan J P de Esch, Rob Leurs
4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H3 Receptor Agonists with in Vivo Central Nervous System Activity. Journal of medicinal chemistry 62 (23) (2019)
Antoni R Blaazer, Abhimanyu K Singh, Erik de Heuvel, Ewald Edink, Kristina M Orrling, Johan J N Veerman, Toine van den Bergh, Chimed Jansen, Erin Balasubramaniam, Wouter J Mooij, Hans Custers, Maarten Sijm, Daniel N A Tagoe, Titilola D Kalejaiye, Jane C Munday, Hermann Tenor, An Matheeussen, Maikel Wijtmans, Marco Siderius, Chris de Graaf, Louis Maes, Harry P de Koning, David S Bailey, Geert Jan Sterk, Iwan J P de Esch, David G Brown, Rob Leurs
Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity. Journal of medicinal chemistry 61 (9) (2018)
Xavier Gómez-Santacana, Sabrina M de Munnik, Prashanna Vijayachandran, Daniel Da Costa Pereira, Jan Paul M Bebelman, Iwan J P de Esch, Henry F Vischer, Maikel Wijtmans, Rob Leurs
Photoswitching the Efficacy of a Small-Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism. Angewandte Chemie (International ed. in English) 57 (36) (2018)