Michael J Waring

ORCID

Publication Activity (10 Years)

Years Active: 2019-2024
Publications (10 Years): 25

Top Venues

Journal of medicinal chemistry

Chemistry (Weinheim an der Bergstrasse, Germany)

Bioconjugate chemistry

Angewandte Chemie (Weinheim an der Bergstrasse, Germany)

Newcastle University

University of Manchester (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Newcastle University

United Kingdom

Professor of Medicinal Chemistry :: Chemistry

AstraZeneca Alderley Park

United Kingdom

Principal Scientist :: Medicinal Chemistry

University of Texas at Austin

United States

Post doctoral researcher :: Chemistry and Biochemistry

Education History

University of Manchester

United Kingdom

PHD :: Chemistry

University of Manchester

United Kingdom

BSC :: Chemistry

Publications

Matthew J Anderson, Thomas P Carton, Catherine L A Salvini, James J Crawford, Garry Pairaudeau, Michael J Waring
Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis. Chemistry (Weinheim an der Bergstrasse, Germany) 30 (21) (2024)
Matthew J Anderson, Thomas P Carton, Catherine L A Salvini, James J Crawford, Garry Pairaudeau, Michael J Waring
Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis. Chemistry (Weinheim an der Bergstrasse, Germany) 30 (21) (2024)
Rachael Pirie, Harriet A Stanway-Gordon, Hannah L Stewart, Kirsty L Wilson, Summer Patton, Jack Tyerman, Daniel J Cole, Katherine Fowler, Michael J Waring
An analysis of the physicochemical properties of oral drugs from 2000 to 2022. RSC medicinal chemistry 15 (9) (2024)
Matthew J Anderson, Thomas P Carton, Catherine L A Salvini, James J Crawford, Garry Pairaudeau, Michael J Waring
Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis. Chemistry (Weinheim an der Bergstrasse, Germany) (2024)
Matthew J Anderson, Thomas P Carton, Catherine L A Salvini, James J Crawford, Garry Pairaudeau, Michael J Waring
Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis. Chemistry (Weinheim an der Bergstrasse, Germany) 30 (21) (2024)
Harriet A Stanway-Gordon, Jake A Odger, Michael J Waring
Development of a Micellar-Promoted Heck Reaction for the Synthesis of DNA-Encoded Libraries. Bioconjugate chemistry (2023)
Harriet A Stanway-Gordon, Jake A Odger, Michael J Waring
Development of a Micellar-Promoted Heck Reaction for the Synthesis of DNA-Encoded Libraries. Bioconjugate chemistry (2023)
Pasquale A Morese, Nahoum Anthony, Michael S Bodnarchuk, Claire Jennings, Mathew P Martin, Richard A Noble, Nicole Phillips, Huw D Thomas, Lan Z Wang, Andrew Lister, Martin E M Noble, Richard A Ward, Stephen R Wedge, Hannah L Stewart, Michael J Waring
Targeting Cytotoxic Agents through EGFR-Mediated Covalent Binding and Release. Journal of medicinal chemistry (2023)
Catherine L A Salvini, Benoit Darlot, Jack Davison, Mathew P Martin, Susan J Tudhope, Shannon Turberville, Akane Kawamura, Martin E M Noble, Stephen R Wedge, James J Crawford, Michael J Waring
Fragment expansion with NUDELs - poised DNA-encoded libraries. Chemical science 14 (31) (2023)
Duncan C Miller, Tristan Reuillon, Lauren Molyneux, Timothy Blackburn, Simon J Cook, Noel Edwards, Jane A Endicott, Bernard T Golding, Roger J Griffin, Ian Hardcastle, Suzannah J Harnor, Amy Heptinstall, Pamela Lochhead, Mathew P Martin, Nick C Martin, Stephanie Myers, David R Newell, Richard A Noble, Nicole Phillips, Laurent Rigoreau, Huw Thomas, Julie A Tucker, Lan-Zhen Wang, Michael J Waring, Ai-Ching Wong, Stephen R Wedge, Martin E M Noble, Celine Cano
Parallel Optimization of Potency and Pharmacokinetics Leading to the Discovery of a Pyrrole Carboxamide ERK5 Kinase Domain Inhibitor. Journal of medicinal chemistry 65 (9) (2022)
Gemma Davison, Mathew P Martin, Shannon Turberville, Selma Dormen, Richard Heath, Amy B Heptinstall, Marie Lawson, Duncan C Miller, Yi Min Ng, James N Sanderson, Ian Hope, Daniel J Wood, Celine Cano, Jane A Endicott, Ian R Hardcastle, Martin E M Noble, Michael J Waring
Mapping Ligand Interactions of Bromodomains BRD4 and ATAD2 with FragLites and PepLites─Halogenated Probes of Druglike and Peptide-like Molecular Interactions. Journal of medicinal chemistry 65 (22) (2022)
Mélanie Uguen, Gemma Davison, Lukas J Sprenger, James H Hunter, Mathew P Martin, Shannon Turberville, Jessica E Watt, Bernard T Golding, Martin E M Noble, Hannah L Stewart, Michael J Waring
Build-Couple-Transform: A Paradigm for Lead-like Library Synthesis with Scaffold Diversity. Journal of medicinal chemistry 65 (16) (2022)
Harriet A Stanway-Gordon, Jessica S Graham, Michael J Waring
On-DNA Transfer Hydrogenolysis and Hydrogenation for the Synthesis of DNA-Encoded Chemical Libraries. Angewandte Chemie (International ed. in English) (2021)
Jessica S Graham, James H Hunter, Michael J Waring
Micellar Buchwald-Hartwig Coupling of Aryl and Heteroarylamines for the Synthesis of DNA-Encoded Libraries. The Journal of organic chemistry 86 (23) (2021)
James H Hunter, Marco Potowski, Harriet A Stanway-Gordon, Andrew Madin, Garry Pairaudeau, Andreas Brunschweiger, Michael J Waring
Functional Group Tolerance of a Micellar on-DNA Suzuki-Miyaura Cross-Coupling Reaction for DNA-Encoded Library Design. The Journal of organic chemistry (2021)
Edwige M H Picazo, Amy B Heptinstall, David M Wilson, Céline Cano, Bernard T Golding, Michael J Waring
Cyclizations and fragmentations in the alkylation of 6-chloro-5-hydroxy-4-aminopyrimidines with aminoalkyl chlorides. Journal of heterocyclic chemistry 58 (4) (2021)
Islam Al-Khawaldeh, Mohammed J Al Yasiri, Gregory G Aldred, Christine Basmadjian, Cinzia Bordoni, Suzannah J Harnor, Amy B Heptinstall, Stephen J Hobson, Claire E Jennings, Shaimaa Khalifa, Honorine Lebraud, Mathew P Martin, Duncan C Miller, Harry J Shrives, João V de Souza, Hannah L Stewart, Max Temple, Huw D Thomas, Jane Totobenazara, Julie A Tucker, Susan J Tudhope, Lan Z Wang, Agnieszka K Bronowska, Celine Cano, Jane A Endicott, Bernard T Golding, Ian R Hardcastle, Ian Hickson, Stephen R Wedge, Elaine Willmore, Martin E M Noble, Michael J Waring
An Alkynylpyrimidine-Based Covalent Inhibitor That Targets a Unique Cysteine in NF-κB-Inducing Kinase. Journal of medicinal chemistry 64 (14) (2021)
Mélanie Uguen, Conghao Gai, Lukas J Sprenger, Hang Liu, Andrew G Leach, Michael J Waring
Microwave-assisted synthesis of 4-oxo-2-butenoic acids by aldol-condensation of glyoxylic acid. RSC advances 11 (48) (2021)
Harriet A Stanway-Gordon, Jessica S Graham, Michael J Waring
On-DNA Transfer Hydrogenolysis and Hydrogenation for the Synthesis of DNA-Encoded Chemical Libraries. Angewandte Chemie (Weinheim an der Bergstrasse, Germany) 134 (3) (2021)
Harriet A Stanway-Gordon, Jessica S Graham, Michael J Waring
On-DNA Transfer Hydrogenolysis and Hydrogenation for the Synthesis of DNA-Encoded Chemical Libraries. Angewandte Chemie (Weinheim an der Bergstrasse, Germany) 134 (3) (2021)
Kirsten McAulay, Emily A Hoyt, Morgan Thomas, Marianne Schimpl, Michael S Bodnarchuk, Hilary J Lewis, Derek Barratt, Deepa Bhavsar, David M Robinson, Michael J Deery, Derek J Ogg, Gonçalo J L Bernardes, Richard A Ward, Michael J Waring, Jason G Kettle
Alkynyl Benzoxazines and Dihydroquinazolines as Cysteine Targeting Covalent Warheads and Their Application in Identification of Selective Irreversible Kinase Inhibitors. Journal of the American Chemical Society 142 (23) (2020)
James H Hunter, Lisa Prendergast, Louis F Valente, Andrew Madin, Garry Pairaudeau, Michael J Waring
High Fidelity Suzuki-Miyaura Coupling for the Synthesis of DNA Encoded Libraries Enabled by Micelle Forming Surfactants. Bioconjugate chemistry 31 (1) (2020)
Alice Douangamath, Daren Fearon, Paul Gehrtz, Tobias Krojer, Petra Lukacik, C David Owen, Efrat Resnick, Claire Strain-Damerell, Anthony Aimon, Péter Ábrányi-Balogh, José Brandão-Neto, Anna Carbery, Gemma Davison, Alexandre Dias, Thomas D Downes, Louise Dunnett, Michael Fairhead, James D Firth, S Paul Jones, Aaron Keeley, György M Keserü, Hanna F Klein, Mathew P Martin, Martin E M Noble, Peter O'Brien, Ailsa J Powell, Rambabu N Reddi, Rachael E Skyner, Matthew Snee, Michael J Waring, Conor Wild, Nir London, Frank von Delft, Martin Austin Walsh
Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease. Nature communications 11 (1) (2020)
Reggie Bosma, Zhiyong Wang, Albert Jelke Kooistra, Nick Bushby, Sebastiaan Kuhne, Jelle van den Bor, Michael J Waring, Chris de Graaf, Iwan J de Esch, Henry F Vischer, Robert J Sheppard, Maikel Wijtmans, Rob Leurs
Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine. Journal of medicinal chemistry 62 (14) (2019)
Daniel J Wood, J Daniel Lopez-Fernandez, Leanne E Knight, Islam Al-Khawaldeh, Conghao Gai, Shengying Lin, Mathew P Martin, Duncan C Miller, Celine Cano, Jane A Endicott, Ian R Hardcastle, Martin E M Noble, Michael J Waring
FragLites-Minimal, Halogenated Fragments Displaying Pharmacophore Doublets. An Efficient Approach to Druggability Assessment and Hit Generation. Journal of medicinal chemistry 62 (7) (2019)

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Publication Activity (10 Years)

Top Topics

Top Venues

Michael J Waring