Peter S Dragovich

ORCID

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 13

Top Venues

Journal of medicinal chemistry

ChemMedChem

Chemical Society reviews

Chemistry (Weinheim an der Bergstrasse, Germany)

This page only lists publications with an associated author ORCID identifier.

Publications

Michael Berlin, Jennifer Cantley, Mark Bookbinder, Elizabeth Bortolon, Fabio Broccatelli, Greg Cadelina, Emily W Chan, Huifen Chen, Xin Chen, Yunxing Cheng, Tommy K Cheung, Kim Davenport, Dean DiNicola, Debbie Gordon, Brian D Hamman, Alicia Harbin, Roy Haskell, Mingtao He, Alison J Hole, Thomas Januario, Philip S Kerry, Stefan G Koenig, Limei Li, Mark Merchant, Inmaculada Pérez-Dorado, Jennifer Pizzano, Connor Quinn, Christopher M Rose, Emma Rousseau, Leofal Soto, Leanna R Staben, Hongming Sun, Qingping Tian, Jing Wang, Weifeng Wang, Crystal S Ye, Xiaofen Ye, Penghong Zhang, Yuhui Zhou, Robert Yauch, Peter S Dragovich
PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models. Journal of medicinal chemistry (2024)
Michael Berlin, Jennifer Cantley, Mark Bookbinder, Elizabeth Bortolon, Fabio Broccatelli, Greg Cadelina, Emily W Chan, Huifen Chen, Xin Chen, Yunxing Cheng, Tommy K Cheung, Kim Davenport, Dean DiNicola, Debbie Gordon, Brian D Hamman, Alicia Harbin, Roy Haskell, Mingtao He, Alison J Hole, Thomas Januario, Philip S Kerry, Stefan G Koenig, Limei Li, Mark Merchant, Inmaculada Pérez-Dorado, Jennifer Pizzano, Connor Quinn, Christopher M Rose, Emma Rousseau, Leofal Soto, Leanna R Staben, Hongming Sun, Qingping Tian, Jing Wang, Weifeng Wang, Crystal S Ye, Xiaofen Ye, Penghong Zhang, Yuhui Zhou, Robert Yauch, Peter S Dragovich
PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models. Journal of medicinal chemistry 67 (2) (2024)
Michael Berlin, Jennifer Cantley, Mark Bookbinder, Elizabeth Bortolon, Fabio Broccatelli, Greg Cadelina, Emily W Chan, Huifen Chen, Xin Chen, Yunxing Cheng, Tommy K Cheung, Kim Davenport, Dean DiNicola, Debbie Gordon, Brian D Hamman, Alicia Harbin, Roy Haskell, Mingtao He, Alison J Hole, Thomas Januario, Philip S Kerry, Stefan G Koenig, Limei Li, Mark Merchant, Inmaculada Pérez-Dorado, Jennifer Pizzano, Connor Quinn, Christopher M Rose, Emma Rousseau, Leofal Soto, Leanna R Staben, Hongming Sun, Qingping Tian, Jing Wang, Weifeng Wang, Crystal S Ye, Xiaofen Ye, Penghong Zhang, Yuhui Zhou, Robert Yauch, Peter S Dragovich
PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models. Journal of medicinal chemistry 67 (2) (2024)
Peter S Dragovich
Degrader-antibody conjugates. Chemical Society reviews 51 (10) (2022)
Peter S Dragovich, Wolfgang Haap, Melinda M Mulvihill, Jean-Marc Plancher, Antonia F Stepan
Small-Molecule Lead-Finding Trends across the Roche and Genentech Research Organizations. Journal of medicinal chemistry 65 (4) (2022)
Peter S Dragovich
Antibody-Drug Conjugates for Immunology. Journal of medicinal chemistry 65 (6) (2022)
Peter S Dragovich, Thomas H Pillow, Robert A Blake, Jack D Sadowsky, Emel Adaligil, Pragya Adhikari, Jinhua Chen, Nicholas Corr, Josefa Dela Cruz-Chuh, Geoffrey Del Rosario, Aaron Fullerton, Steven J Hartman, Fan Jiang, Susan Kaufman, Tracy Kleinheinz, Katherine R Kozak, Liling Liu, Ying Lu, Melinda M Mulvihill, Jeremy M Murray, Aimee O'Donohue, Rebecca K Rowntree, William S Sawyer, Leanna R Staben, John Wai, Jian Wang, BinQing Wei, Wentao Wei, Zijin Xu, Hui Yao, Shang-Fan Yu, Donglu Zhang, Hongyan Zhang, Shenhua Zhang, Yongxin Zhao, Hao Zhou, Xiaoyu Zhu
Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 2: Improvement of In Vitro Antiproliferation Activity and In Vivo Antitumor Efficacy. Journal of medicinal chemistry 64 (5) (2021)
Peter S Dragovich, Thomas H Pillow, Robert A Blake, Jack D Sadowsky, Emel Adaligil, Pragya Adhikari, Sunil Bhakta, Nicole Blaquiere, Jinhua Chen, Josefa Dela Cruz-Chuh, Karen E Gascoigne, Steven J Hartman, Mingtao He, Susan Kaufman, Tracy Kleinheinz, Katherine R Kozak, Liang Liu, Liling Liu, Qi Liu, Ying Lu, Fanwei Meng, Melinda M Mulvihill, Aimee O'Donohue, Rebecca K Rowntree, Leanna R Staben, Steven T Staben, John Wai, Jian Wang, BinQing Wei, Catherine Wilson, Jianfeng Xin, Zijin Xu, Hui Yao, Donglu Zhang, Hongyan Zhang, Hao Zhou, Xiaoyu Zhu
Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1: Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties. Journal of medicinal chemistry 64 (5) (2021)
Leanna R Staben, Jinhua Chen, Josefa Dela Cruz-Chuh, Geoff Del Rosario, Mary Ann Go, Jun Guo, S Cyrus Khojasteh, Katherine R Kozak, Guangmin Li, Carl Ng, Gail D Lewis Phillips, Thomas H Pillow, Rebecca K Rowntree, John Wai, BinQing Wei, Keyang Xu, Zijin Xu, Shang-Fan Yu, Donglu Zhang, Peter S Dragovich
Systematic Variation of Pyrrolobenzodiazepine (PBD)-Dimer Payload Physicochemical Properties Impacts Efficacy and Tolerability of the Corresponding Antibody-Drug Conjugates. Journal of medicinal chemistry 63 (17) (2020)
Dian Su, Jinhua Chen, Ely Cosino, Josefa Dela Cruz-Chuh, Helen Davis, Geoffrey Del Rosario, Isabel Figueroa, Leanne Goon, Jintang He, Amrita V Kamath, Surinder Kaur, Katherine R Kozak, Jeffrey Lau, Donna Lee, M Violet Lee, Douglas Leipold, Luna Liu, Peter Liu, Guo-Liang Lu, Chris Nelson, Carl Ng, Thomas H Pillow, Paul Polakis, Andrew G Polson, Rebecca K Rowntree, Ola Saad, Brian Safina, Nicola J Stagg, Moana Tercel, Richard Vandlen, Breanna S Vollmar, John Wai, Tao Wang, BinQing Wei, Keyang Xu, Juanjuan Xue, Zijin Xu, Gang Yan, Hui Yao, Shang-Fan Yu, Donglu Zhang, Fiona Zhong, Peter S Dragovich
Antibody-Drug Conjugates Derived from Cytotoxic seco-CBI-Dimer Payloads Are Highly Efficacious in Xenograft Models and Form Protein Adducts In Vivo. Bioconjugate chemistry 30 (5) (2019)
Thomas H Pillow, Pragya Adhikari, Robert A Blake, Jinhua Chen, Geoffrey Del Rosario, Gauri Deshmukh, Isabel Figueroa, Karen E Gascoigne, Amrita V Kamath, Susan Kaufman, Tracy Kleinheinz, Katherine R Kozak, Brandon Latifi, Douglas D Leipold, Chun Sing Li, Ruina Li, Melinda M Mulvihill, Aimee O'Donohue, Rebecca K Rowntree, Jack D Sadowsky, John Wai, Xinxin Wang, Cong Wu, Zijin Xu, Hui Yao, Shang-Fan Yu, Donglu Zhang, Richard Zang, Hongyan Zhang, Hao Zhou, Xiaoyu Zhu, Peter S Dragovich
Antibody Conjugation of a Chimeric BET Degrader Enables in vivo Activity. ChemMedChem 15 (1) (2019)
Peter S Dragovich, Robert A Blake, Chunjiao Chen, Jinhua Chen, Josefa Chuh, Willem den Besten, Fang Fan, Aimee Fourie, Steven J Hartman, Changrong He, Jintang He, Ellen Rei Ingalla, Katherine R Kozak, Steven R Leong, Jiawei Lu, Yong Ma, Lingyao Meng, Michelle Nannini, Jason Oeh, Rachana Ohri, Gail Lewis Phillips, Thomas H Pillow, Rebecca K Rowntree, Deepak Sampath, Richard Vandlen, Breanna Vollmar, John Wai, Ingrid E Wertz, Keyang Xu, Zijin Xu, Donglu Zhang
Conjugation of Indoles to Antibodies through a Novel Self-Immolating Linker. Chemistry (Weinheim an der Bergstrasse, Germany) 24 (19) (2018)
Zhonghua Pei, Chunjiao Chen, Jinhua Chen, Josefa Dela Cruz-Chuh, Reginald Delarosa, Yuzhong Deng, Aimee Fourie-O'Donohue, Isabel Figueroa, Jun Guo, Weiwei Jin, S Cyrus Khojasteh, Katherine R Kozak, Brandon Latifi, James Lee, Guangmin Li, Eva Lin, Liling Liu, Jiawei Lu, Scott Martin, Carl Ng, Trung Nguyen, Rachana Ohri, Gail Lewis Phillips, Thomas H Pillow, Rebecca K Rowntree, Nicola J Stagg, David Stokoe, Sheila Ulufatu, Vishal A Verma, John Wai, Jing Wang, Keyang Xu, Zijin Xu, Hui Yao, Shang-Fan Yu, Donglu Zhang, Peter S Dragovich
Exploration of Pyrrolobenzodiazepine (PBD)-Dimers Containing Disulfide-Based Prodrugs as Payloads for Antibody-Drug Conjugates. Molecular pharmaceutics 15 (9) (2018)

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Publication Activity (10 Years)

Top Topics

Top Venues

Peter S Dragovich