Simon J F Macdonald (S J F Macdonald, Simon Jf Macdonald)

ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 12

Top Venues

Journal of medicinal chemistry

Nature reviews. Drug discovery

Future medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Panayiotis A Procopiou, John Barrett, Matthew H J Crawford, Richard J D Hatley, Ashley P Hancock, John M Pritchard, James E Rowedder, Royston C B Copley, Robert J Slack, Steven L Sollis, Lee R Thorp, Rhys A Lippa, Simon J F Macdonald, Tim N Barrett
Discovery and Development of Highly Potent and Orally Bioavailable Nonpeptidic α v β 6 Integrin Inhibitors. Journal of medicinal chemistry (2024)
Simon J F Macdonald
Medicinal chemistry in big pharma has a gender diversity problem. Future medicinal chemistry 14 (19) (2022)
Jennifer M Clark, Fernando Salgado-Polo, Simon J F Macdonald, Tim N Barrett, Anastassis Perrakis, Craig J Jamieson
Structure-Based Design of a Novel Class of Autotaxin Inhibitors Based on Endogenous Allosteric Modulators. Journal of medicinal chemistry 65 (8) (2022)
Richard J D Hatley, Steve P McLachlan, Kathleen Baster, Lucy C Gelder, Simon J F Macdonald
How Diverse Is Medicinal Chemistry? Insights into Race, Ethnicity, Origin, Gender, and Geography. Journal of medicinal chemistry 65 (1) (2021)
R J Slack, Simon J F Macdonald, James A Roper, R Gisli Jenkins, Richard J D Hatley
Emerging therapeutic opportunities for integrin inhibitors. Nature reviews. Drug discovery (2021)
Richard J D Hatley, Panayiotis A Procopiou, Steven P McLachlan, Laura E Westendorf, Nicholas A Meanwell, William R Ewing, Simon J F Macdonald
Writing Your Next Medicinal Chemistry Article: Journal Bibliometrics and Guiding Principles for Industrial Authors. Journal of medicinal chemistry 63 (23) (2020)
Niall A Anderson, Sebastien Campos, Sharon Butler, Royston C B Copley, Ian Duncan, Stephen Harrison, Joelle Le, Rosemary Maghames, Aleix Pastor-Garcia, John M Pritchard, James E Rowedder, Claire E Smith, Jack Thomas, Giovanni Vitulli, Simon J F Macdonald
Discovery of an Orally Bioavailable Pan αv Integrin Inhibitor for Idiopathic Pulmonary Fibrosis. Journal of medicinal chemistry 62 (19) (2019)
Tim N Barrett, Jonathan A Taylor, Daniel Barker, Panayiotis A Procopiou, James D F Thompson, John Barrett, Joelle Le, Sean M Lynn, Peter Pogany, Cassie Pratley, John M Pritchard, James A Roper, James E Rowedder, Robert J Slack, Giovanni Vitulli, Simon J F Macdonald, William J Kerr
Profile of a Highly Selective Quaternized Pyrrolidine Betaine αvβ6 Integrin Inhibitor-(3S)-3-(3-(3,5-Dimethyl-1H-pyrazol-1-yl)phenyl)-4-((1S and 1R,3R)-1-methyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-ium-1-yl)butanoate Synthesized by Stereoselective Methylation. Journal of medicinal chemistry 62 (16) (2019)
Panayiotis A Procopiou, Niall A Anderson, John Barrett, Tim N Barrett, Matthew H J Crawford, Brendan J Fallon, Ashley P Hancock, Joelle Le, Seble Lemma, Richard P Marshall, Josie Morrell, John M Pritchard, James E Rowedder, Paula Saklatvala, Robert J Slack, Steven L Sollis, Colin J Suckling, Lee R Thorp, Giovanni Vitulli, Simon J F Macdonald
Discovery of ( S)-3-(3-(3,5-Dimethyl-1 H-pyrazol-1-yl)phenyl)-4-(( R)-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-yl)butanoic Acid, a Nonpeptidic αvβ6 Integrin Inhibitor for the Inhaled Treatment of Idiopathic Pulmonary Fibrosis. Journal of medicinal chemistry 61 (18) (2018)
Willem-Jan Keune, Frances Potjewyd, Tatjana Heidebrecht, Fernando Salgado-Polo, Simon J F Macdonald, Lakshman Chelvarajan, Ahmed Abdel Latif, Sony Soman, Andrew J Morris, Allan J B Watson, Craig J Jamieson, Anastassis Perrakis
Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators. Journal of medicinal chemistry 60 (5) (2017)
Elena Sandoval, María José Lafuente-Monasterio, María J Almela, Pablo Castañeda, María Belén Jiménez Díaz, María S Martínez-Martínez, Jaume Vidal, Íñigo Angulo-Barturen, Paul Bamborough, Jeremy Burrows, Nicholas Cammack, María J Chaparro, José M Coterón, Cristina de Cozar, Benigno Crespo, Beatriz Díaz, Gerard Drewes, Esther Fernández, Santiago Ferrer-Bazaga, María Teresa Fraile, Francisco J Gamo, Sonja Ghidelli-Disse, Rubén Gómez, John Haselden, Sophie Huss, María Luisa León, Jaime de Mercado, Simon J F Macdonald, José Ignacio Martín Hernando, Sara Prats, Margarita Puente, Anne Rodríguez, Juan C de la Rosa, Lourdes Rueda, Carolyn Selenski, Paul Willis, David M Wilson, Michael Witty, Felix Calderon
The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold. Journal of medicinal chemistry 60 (16) (2017)
Thomas McInally, Simon J F Macdonald
Unusual Undergraduate Training in Medicinal Chemistry in Collaboration between Academia and Industry. Journal of medicinal chemistry 60 (19) (2017)

Simon J F Macdonald.css-eqlu8i{font-size:small;padding-left:4px;} (S J F Macdonald, Simon Jf Macdonald)

Publication Activity (10 Years)

Top Topics

Top Venues

Simon J F Macdonald (S J F Macdonald, Simon Jf Macdonald)