William J Kerr

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2016-2023
Publications (10 Years): 13

Top Topics

Reduced Graphene Oxide

Transition Metal

Tyrosine Kinase

Top Venues

Journal of medicinal chemistry

Angewandte Chemie (International ed. in English)

Chemical science

Journal of labelled compounds & radiopharmaceuticals

This page only lists publications with an associated author ORCID identifier.

Publications

Erin Bradley, Lucia Fusani, Chun-Wa Chung, Peter D Craggs, Emmanuel H Demont, Philip G Humphreys, Darren J Mitchell, Alex Phillipou, Inmaculada Rioja, Rishi R Shah, Christopher R Wellaway, Rab K Prinjha, David S Palmer, William J Kerr, Marc Reid, Ian D Wall, Rosa Cookson
Structure-Guided Design of a Domain-Selective Bromodomain and Extra Terminal N-Terminal Bromodomain Chemical Probe. Journal of medicinal chemistry (2023)
Callum G J Hall, Helen F Sneddon, Peter Pogány, David M Lindsay, William J Kerr
Experimental and computational insights into the mechanism of the copper(i)-catalysed sulfonylative Suzuki-Miyaura reaction. Chemical science 14 (24) (2023)
Elliot Davenport, Daniela E Negru, Geoff Badman, David M Lindsay, William J Kerr
Robust and General Late-Stage Methylation of Aryl Chlorides: Application to Isotopic Labeling of Drug-like Scaffolds. ACS catalysis 13 (17) (2023)
Paul Shaw, Storm J Hassell-Hart, Gayle E Douglas, Andrew G Malcolm, Alan R Kennedy, Gemma V White, Laura C Paterson, William J Kerr
Oxygenated Cyclopentenones via the Pauson-Khand Reaction of Silyl Enol Ether Substrates. Organic letters 24 (14) (2022)
William J Kerr, Gary J Knox, Marc Reid, Tell Tuttle
Catalyst design in C-H activation: a case study in the use of binding free energies to rationalise intramolecular directing group selectivity in iridium catalysis. Chemical science 12 (19) (2021)
Christopher R Wellaway, Paul Bamborough, Sharon G Bernard, Chun-Wa Chung, Peter D Craggs, Leanne Cutler, Emmanuel H Demont, John P Evans, Laurie Gordon, Bhumika Karamshi, Antonia J Lewis, Matthew J Lindon, Darren J Mitchell, Inmaculada Rioja, Peter E Soden, Simon Taylor, Robert J Watson, Rob Willis, James M Woolven, Beata S Wyspiańska, William J Kerr, Rab K Prinjha
Structure-Based Design of a Bromodomain and Extraterminal Domain (BET) Inhibitor Selective for the N-Terminal Bromodomains That Retains an Anti-inflammatory and Antiproliferative Phenotype. Journal of medicinal chemistry 63 (17) (2020)
William J Kerr, Gary J Knox, Laura C Paterson
Recent advances in iridium(I) catalysis towards directed hydrogen isotope exchange. Journal of labelled compounds & radiopharmaceuticals 63 (6) (2020)
Adele E Queen, David Hesk, David M Lindsay, William J Kerr, Kenneth Rehder, Tim Fennell, S Wayne Mascarella, Desong Zhong, Scott Runyon
Synthesis of [3 H] and [14 C]genipin. Journal of labelled compounds & radiopharmaceuticals 63 (4) (2020)
Tim N Barrett, Jonathan A Taylor, Daniel Barker, Panayiotis A Procopiou, James D F Thompson, John Barrett, Joelle Le, Sean M Lynn, Peter Pogany, Cassie Pratley, John M Pritchard, James A Roper, James E Rowedder, Robert J Slack, Giovanni Vitulli, Simon J F Macdonald, William J Kerr
Profile of a Highly Selective Quaternized Pyrrolidine Betaine αvβ6 Integrin Inhibitor-(3S)-3-(3-(3,5-Dimethyl-1H-pyrazol-1-yl)phenyl)-4-((1S and 1R,3R)-1-methyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-ium-1-yl)butanoate Synthesized by Stereoselective Methylation. Journal of medicinal chemistry 62 (16) (2019)
Christopher P Tinworth, Hannah Lithgow, Lars Dittus, Zuni I Bassi, Sophie E Hughes, Marcel Muelbaier, Han Dai, Ian E D Smith, William J Kerr, Glenn A Burley, Marcus Bantscheff, John D Harling
PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding. ACS chemical biology 14 (3) (2019)
Jason D Williams, William J Kerr, Stuart G Leach, David M Lindsay
A Practical and General Amidation Method from Isocyanates Enabled by Flow Technology. Angewandte Chemie (International ed. in English) 57 (37) (2018)
William J Kerr, Marc Reid, Tell Tuttle
Iridium-Catalyzed Formyl-Selective Deuteration of Aldehydes. Angewandte Chemie (International ed. in English) 56 (27) (2017)
William J Kerr, Richard J Mudd, Jack A Brown
Iridium(I) N-Heterocyclic Carbene (NHC)/Phosphine Catalysts for Mild and Chemoselective Hydrogenation Processes. Chemistry (Weinheim an der Bergstrasse, Germany) 22 (14) (2016)